Bromide

Bromide

SCHEMBL7904291

Br.N=C(N)c1ccc(O)c(F)c1

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F12 P00748 1/20 0.47
LMNA P02545 2/20 0.46
PRSS1 P07477 5/20 0.45
PRSS3 P35030 3/20 0.45
PRSS2 P07478 2/20 0.45
F2 P00734 4/20 0.44
PLAU P00749 3/20 0.44
PLG P00747 3/20 0.44
KLK1 P06870 2/20 0.44
KLKB1 P03952 1/20 0.44
KDM1A O60341 1/20 0.44
KLK5 Q9Y337 1/20 0.43
SNCA P37840 1/20 0.43
KDM4E B2RXH2 1/20 0.43
HSD17B10 Q99714 1/20 0.43
F10 P00742 1/20 0.42
PLAT P00750 1/20 0.42
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
MASP2 O00187 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12581536 0.98 F12 (0.48) F12LMNAPRSS1PRSS3PRSS2
Hydrochloric Acid SCHEMBL7913049 0.96 F12 (0.47) F12LMNAPRSS1PRSS3PRSS2
Hydrochloric Acid SCHEMBL22974828 0.94 F12 (0.46) F12LMNAPRSS1PRSS3PRSS2
Trifluoroacetic Acid SCHEMBL13269627 0.84 KLK1 (0.47) LMNAPRSS1F2KLK1KLK5
SCHEMBL1713947 0.82 LMNA (0.61) LMNAPLAUKDM4EHSD17B10ESR1
SCHEMBL1262883 0.80 CES2 (0.54) F12LMNAPRSS1PRSS3PRSS2
Hydrochloric Acid SCHEMBL3515941 0.78 LMNA (0.52) F12LMNAPRSS1PRSS3PRSS2
SCHEMBL9314470 0.78 LMNA (0.54) F12LMNAPRSS1PRSS3PRSS2
SCHEMBL22995847 0.77 SNCA (0.44) LMNAKDM1ASNCAKDM4EHSD17B10
SCHEMBL1061714 0.77 LCK (0.53) LMNAKDM1ASNCAKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1135450-A1 CHIRAL LIQUID CRYSTAL COMPOUNDS HAVING A FLUORINATED TERMINAL PORTION MINNESOTA MINING AND MANUFACTURING COMPANY (US) 2001-09-26 EP disclosed
US-6139924-A CONTAINING A PYRIMIDINE RING 3M INNOVATIVE PROPERTIES COMPANY (US) 2000-10-31 US disclosed
WO-2000031210-A1 CHIRAL LIQUID CRYSTAL COMPOUNDS HAVING A FLUORINATED TERMINAL PORTION MINNESOTA MINING AND MANUFACTURING COMPANY (US) 2000-06-02 WO disclosed
US-5928562-A HAVING EXTENDED HYDROCARBON ETHER GROUP ADJACENT TO A TERMINAL FLUOROALKYL OR FLUOROETHER GROUP; LOW VISCOSITY; HIGH SPEED RESPONSE; BRIGHTNESS; COMMPATIBILITY; DISPLAYS MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1999-07-27 US disclosed