SCHEMBL7904785

SCHEMBL7904785

CSc1nc(NNC(=O)c2cccnc2)cc(Oc2ccccc2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.46
HTT P42858 2/20 0.46
MEN1 O00255 2/20 0.46
ALDH1A1 P00352 2/20 0.43
ALOX15 P16050 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
LMNA P02545 3/20 0.43
TSHR P16473 3/20 0.43
NPSR1 Q6W5P4 1/20 0.43
GRM5 P41594 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
MAPT P10636 2/20 0.41
GAA P10253 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
CYP3A4 P08684 1/20 0.41
ALPL P05186 1/20 0.41
ALPI P09923 1/20 0.41
ALPG P10696 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6624562 0.90 MEN1 (0.53) KMT2AHTTMEN1ALDH1A1L3MBTL1
SCHEMBL6627389 0.84 MEN1 (0.54) KMT2AHTTMEN1LMNATSHR
SCHEMBL6624257 0.78 HTT (0.47) KMT2AHTTMEN1ALDH1A1ALOX15
SCHEMBL6628004 0.78 MEN1 (0.47) KMT2AHTTMEN1ALDH1A1L3MBTL1
SCHEMBL6624715 0.76 HTT (0.46) KMT2AHTTMEN1ALDH1A1ALOX15
SCHEMBL6625095 0.73 LMNA (0.44) KMT2AHTTMEN1ALDH1A1ALOX15
SCHEMBL7799660 0.70 HTT (0.81) KMT2AHTTMEN1ALDH1A1L3MBTL1
SCHEMBL6627858 0.70 LMNA (0.45) KMT2AHTTMEN1ALDH1A1ALOX15
SCHEMBL6625937 0.69 NPC1 (0.42) KMT2AHTTMEN1ALDH1A1L3MBTL1
SCHEMBL11832072 0.68 PTGS2 (0.68) ALDH1A1LMNAGAACYP3A4ALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6222035-B1 AS ADENOSINE A.SUB.2A RECEPTOR ANTAGONISTS AND ARE USEFUL FOR THERAPY OR OR PROPHYLAXIS OF VARIOUS DISEASES INDUCED BY HYPERACTIVITY OF ADENOSINE A.SUB.2A RECEPTORS SUCH AS PARKINSON'S DISEASE, SENILE DEMENTIA OR DEPRESSION KYOWA HAKKO KOGYO CO., LTD. (JP) 2001-04-24 US disclosed
EP-0976753-A1 [1,2,4]TRIAZOLO[1,5-c]PYRIMIDINE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 2000-02-02 EP disclosed