SCHEMBL790546

SCHEMBL790546

O=C1OCC(COCc2ccccc2)C1F

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.46
TAAR1 Q96RJ0 1/20 0.46
LMNA P02545 1/20 0.46
CYP3A4 P08684 4/20 0.41
TSHR P16473 2/20 0.41
MAPT P10636 2/20 0.41
CYP2C19 P33261 2/20 0.41
FKBP1A P62942 1/20 0.38
AKT1 P31749 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18302831 0.82 CYP19A1 (0.49) CYP19A1TAAR1LMNACYP3A4TSHR
SCHEMBL24286799 0.82 CYP19A1 (0.49) CYP19A1TAAR1LMNACYP3A4TSHR
SCHEMBL20993237 0.82 CYP19A1 (0.49) CYP19A1TAAR1LMNACYP3A4TSHR
SCHEMBL5725152 0.78 TAAR1 (0.50) CYP19A1TAAR1LMNACYP3A4TSHR
SCHEMBL599776 0.77 LMNA (0.46) TAAR1LMNATSHRAKT1
SCHEMBL599240 0.77 LMNA (0.46) TAAR1LMNATSHRAKT1
SCHEMBL599775 0.77 LMNA (0.46) TAAR1LMNATSHRAKT1
SCHEMBL5112138 0.74 CYP19A1 (0.47) CYP19A1TAAR1LMNACYP3A4TSHR
SCHEMBL30959376 0.73 CYP19A1 (0.52) CYP19A1TAAR1LMNACYP3A4TSHR
SCHEMBL16397855 0.72 TAAR1 (0.50) CYP19A1TAAR1LMNATSHRFKBP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616080-A1 2' -FLUORO SUBSTITUTED CARBA-NUCLEOSIDE ANALOGS FOR ANTIVIRAL TREATMENT Gilead Sciences, Inc. (US) 2013-07-24 EP disclosed
WO-2012037038-A1 2' -FLUORO SUBSTITUTED CARBA-NUCLEOSIDE ANALOGS FOR ANTIVIRAL TREATMENT GILEAD SCIENCES, INC. (US) 2012-03-22 WO disclosed