Pyrene

Pyrene

SCHEMBL7907123

C(=C/c1ccccc1)\c1ccccc1.c1cc2ccc3cccc4ccc(c1)c2c34

nearest known ligand 0.60

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RELA Q04206 1/20 0.60
ALDH1A1 P00352 4/20 0.58
HPGD P15428 3/20 0.58
CYP3A4 P08684 2/20 0.58
TSHR P16473 2/20 0.58
CYP1A2 P05177 2/20 0.58
HSD17B10 Q99714 2/20 0.58
CYP1A1 P04798 1/20 0.58
CYP1B1 Q16678 1/20 0.58
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
KDM4E B2RXH2 2/20 0.52
PKM P14618 2/20 0.52
LMNA P02545 1/20 0.52
MAOB P27338 3/20 0.50
NFE2L2 Q16236 3/20 0.48
CYP19A1 P11511 2/20 0.48
MAOA P21397 2/20 0.48
GRM4 Q14833 2/20 0.47
MEN1 O00255 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyrene SCHEMBL7907124 1.00 RELA (0.60) RELAALDH1A1HPGDCYP3A4TSHR
Pyrene SCHEMBL27498377 0.86 ALDH1A1 (0.48) RELAALDH1A1HPGDCYP3A4TSHR
Pyrene SCHEMBL27594669 0.86 CYP1B1 (0.48) RELAALDH1A1HPGDCYP3A4TSHR
(Z)-1,2-Diphenylethene SCHEMBL27485869 0.85 ALDH1A1 (0.54) RELAALDH1A1HPGDCYP3A4TSHR
SCHEMBL131580 0.84 RELA (0.46) RELAALDH1A1HPGDCYP3A4TSHR
SCHEMBL31550572 0.84 RELA (0.46) RELAALDH1A1HPGDCYP3A4TSHR
SCHEMBL131581 0.84 RELA (0.46) RELAALDH1A1HPGDCYP3A4TSHR
SCHEMBL31236793 0.81 CYP1A2 (0.50) RELAALDH1A1HPGDCYP1A2HSD17B10
Pyrene SCHEMBL9716948 0.80 ALDH1A1 (0.67) RELAALDH1A1HPGDCYP3A4TSHR
Pyrene SCHEMBL4936826 0.80 ALDH1A1 (0.67) RELAALDH1A1HPGDCYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6218108-B1 NUCLEOSIDE DERIVATIVE COMPRISING PYRENE, ANTHRACENE, PHENANTHRENE, STILBENE, TETRACENE OR PENTACENE JOINED TO THE C-1 ATOM OF A RIBOSE OR DEOXYRIBOSE SUGAR; PROBES FOR FLUORESCENT IN SITU HYBRIDIZATION RESEARCH CORPORATION TECHNOLOGIES, INC. 2001-04-17 US disclosed
US-6140480-A ADDUCT OF HOFFER'S CHLOROSUGAR COMPRISING AN ORGANOCADMIUM OR ORGANOZINC DERIVATIVE OF PYRENE, ANTHRACENE, PHENANTHRENE, STILBENE, TETRACENE, OR PENTACENE COUPLED TO THE C1 POSITION; FLUORESCENT PROBES RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 2000-10-31 US disclosed