SCHEMBL7907148

SCHEMBL7907148

Cc1cccc(-c2ccc(C)nc2N)n1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.58
CCR8 P51685 1/20 0.58
NOS3 P29474 1/20 0.48
NOS2 P35228 1/20 0.48
TGFBR1 P36897 14/20 0.44
CYP2A6 P11509 1/20 0.42
METAP2 P50579 1/20 0.42
NSD2 O96028 1/20 0.37
G6PD P11413 1/20 0.37
DNMT1 P26358 1/20 0.37
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23888704 0.79 CCR1 (0.52) CCR1CCR8NOS3NOS2TGFBR1
SCHEMBL7910798 0.79 KDM4E (0.46) CCR1CCR8TGFBR1
SCHEMBL3723641 0.76 CCR1 (0.58) CCR1CCR8NOS3NOS2TGFBR1
SCHEMBL7911485 0.76 CDK2 (0.41) NOS3NOS2TGFBR1
SCHEMBL8101860 0.76 CCR1 (0.52) CCR1CCR8NOS3NOS2TGFBR1
SCHEMBL995546 0.76 CCR1 (0.52) CCR1CCR8NOS3NOS2TGFBR1
SCHEMBL30511194 0.75 CCR1 (1.00) CCR1CCR8NOS3NOS2TGFBR1
SCHEMBL196966 0.75 CCR1 (1.00) CCR1CCR8NOS3NOS2TGFBR1
SCHEMBL29388304 0.75 CCR1 (1.00) CCR1CCR8NOS3NOS2TGFBR1
SCHEMBL5687521 0.74 CCR1 (0.50) CCR1CCR8NOS3NOS2TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063663-A1 N-{[(IR,4S,6R-3-(2-PYRIDINYLCARBONYL)-3-AZABICYCLO [4.1.0]HEPT-4-YL] METHYL}-2-HETEROARYLAMINE DERIVATIVES AND USES THEREOF GLAXO GROUP LIMITED (GB) 2010-06-10 WO disclosed