SCHEMBL7908573

SCHEMBL7908573

CSc1nc(N)n(-c2nnc(-c3cccc(OCCCN(C)C)c3)s2)n1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.49
KDM4E B2RXH2 1/20 0.45
NOTUM Q6P988 1/20 0.42
CHEK2 O96017 1/20 0.38
HDAC1 Q13547 6/20 0.38
HDAC2 Q92769 6/20 0.38
HDAC8 Q9BY41 3/20 0.38
HDAC6 Q9UBN7 3/20 0.38
LSS P48449 1/20 0.37
TNK2 Q07912 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
CXCR1 P25024 1/20 0.36
ADORA2A P29274 1/20 0.36
DCK P27707 1/20 0.35
HCRTR1 O43613 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7905959 0.99 SMN1; SMN2 (0.48) SMN1; SMN2KDM4ENOTUMCHEK2HDAC1
SCHEMBL7905739 0.95 SMN1; SMN2 (0.47) SMN1; SMN2KDM4ENOTUMHDAC1HDAC2
SCHEMBL7905953 0.89 RAB9A (0.45) SMN1; SMN2KDM4ELSSHRH3CXCR1
SCHEMBL7903925 0.89 SMN1; SMN2 (0.51) SMN1; SMN2KDM4ENOTUMHDAC1HDAC2
Hydrochloric Acid SCHEMBL7908541 0.89 RAB9A (0.44) SMN1; SMN2KDM4ELSSHRH3CXCR1
SCHEMBL7896538 0.84 RAB9A (0.43) SMN1; SMN2KDM4ETNK2HRH3ADORA2A
SCHEMBL7896441 0.82 HTR1B (0.37) KDM4ELSSHRH3
Hydrochloric Acid SCHEMBL7903914 0.81 HTR1B (0.36) KDM4ELSSHRH3
SCHEMBL7896418 0.77 RAB9A (0.46) SMN1; SMN2KDM4EHDAC1HDAC2HDAC6
SCHEMBL7905806 0.77 HTR7 (0.40) SMN1; SMN2KDM4EADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191152-B1 CARDIOVASCULAR DISORDERS, NERVOUS SYSTEM DISORDERS EGIS GYÓGYSZERGYAR RT. (HU) 2001-02-20 US claimed
US-6191152-B1 CARDIOVASCULAR DISORDERS, NERVOUS SYSTEM DISORDERS EGIS GYÓGYSZERGYAR RT. (HU) 2001-02-20 US disclosed
EP-0958294-A1 2-(1,2,4-TRIAZOLE-1-YL)-1,3,4-THIADIAZOLE DERIVATIVES HAVING AN EFFECT ON THE C.N.S. AND THE HEART EGIS GYOGYSZERGYAR (HU) 1999-11-24 EP disclosed
WO-1998030561-A1 2-(1,2,4-TRIAZOLE-1-YL)-1,3,4-THIADIAZOLE DERIVATIVES HAVING AN EFFECT ON THE C.N.S. AND THE HEART EGIS Gyógyszergyár Rt. (HU) 1998-07-16 WO disclosed