SCHEMBL7908816

SCHEMBL7908816

O=C(O)CC[C@H](Cl)c1ccccc1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.43
ALDH1A1 P00352 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP1A2 P05177 1/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.42
CPA3 P15088 1/20 0.41
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
GAA P10253 1/20 0.38
MAPK1 P28482 2/20 0.37
KDM4E B2RXH2 1/20 0.37
TP53 P04637 1/20 0.37
GLA P06280 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
HPGD P15428 1/20 0.37
ALOX12 P18054 1/20 0.37
NFKB1 P19838 1/20 0.37
APEX1 P27695 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7908812 1.00 HTT (0.43) HTTALDH1A1CYP2D6CYP1A2TSHR
SCHEMBL27336117 0.80 HTT (0.41) HTTALDH1A1CYP2C19TP53CYSLTR2
SCHEMBL7907656 0.79 ALDH1A1 (0.42) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL7911091 0.79 ALDH1A1 (0.42) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL7907662 0.79 ALDH1A1 (0.42) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL20656719 0.77 HTT (0.46) HTTALDH1A1CYP2C19CYP3A4CYP26A1
SCHEMBL1132531 0.76 CYP2D6 (0.48) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL7910713 0.76 CYP2D6 (0.48) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL7914353 0.76 FFAR1 (0.40) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL11827355 0.76 ALDH1A1 (0.41) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211234-B1 BENZONITRILE COMPOUNDS WITH ETHER AND SULFIDE GROUPS WITH CARBOXY ACID RHONE-POULENC RORER LIMITED (GB) 2001-04-03 US disclosed
EP-0728128-B1 SUBSTITUTED PHENYL COMPOUNDS RHONE POULENC RORER LTD (GB) 1998-09-16 EP disclosed
EP-0728128-A1 SUBSTITUTED PHENYL COMPOUNDS RHONE-POULENC RORER LIMITED (GB) 1996-08-28 EP disclosed
WO-1995013262-A1 SUBSTITUTED PHENYL COMPOUNDS RHONE-POULENC RORER LIMITED (GB) 1995-05-18 WO disclosed