SCHEMBL7908853

SCHEMBL7908853

NNC(=O)[C@H](CCO)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.56
ALDH1A1 P00352 2/20 0.44
GAA P10253 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
EPHX1 P07099 1/20 0.43
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
KCNQ2 O43526 1/20 0.41
MAPT P10636 1/20 0.41
HDAC1 Q13547 4/20 0.40
HDAC7 Q8WUI4 4/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7908761 1.00 CTSD (0.56) CTSDALDH1A1GAASMN1; SMN2EPHX1
SCHEMBL7908764 1.00 CTSD (0.56) CTSDALDH1A1GAASMN1; SMN2EPHX1
SCHEMBL29873777 0.85 CTSD (0.60) CTSDEPHX1KCNQ2MAPTHDAC1
SCHEMBL8113733 0.84 CTSD (0.55) CTSDALDH1A1SMN1; SMN2KCNQ2MAPT
SCHEMBL7906036 0.83 ALDH1A1 (0.44) CTSDALDH1A1GAACNR2HDAC1
SCHEMBL1533332 0.83 ALDH1A1 (0.44) CTSDALDH1A1GAACNR2HDAC1
SCHEMBL7908914 0.83 ALDH1A1 (0.44) CTSDALDH1A1GAACNR2HDAC1
Hydrochloric Acid SCHEMBL908853 0.83 CTSD (0.53) CTSDALDH1A1EPHX1CNR1CNR2
SCHEMBL9702168 0.81 CTSD (0.51) CTSDALDH1A1SMN1; SMN2EPHX1MAPT
SCHEMBL908825 0.81 CTSD (0.51) CTSDSMN1; SMN2EPHX1CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207862-B1 PRECURSORS ARE CHIRAL 4-HYDROXYCARBOXAMIDES, 4-HYDROXYHYDROXAMIC ACIDS, OR 4-HYDROXYHYDRAZIDES PRODUCED FROM GAMMA-LACTONES, WHICH IN TURN ARE DERIVED FROM 1,4-DIOLS BY STEREOSELECTIVE OXIDATION, BIOCATALYTICS, INC. 2001-03-27 US disclosed
WO-1999032649-A1 METHODS AND PRECURSORS FOR THE PRODUCTION OF CHIRAL 1,3-AMINOALCOHOLS BIOCATALYTICS, INC. (US) 1999-07-01 WO disclosed
US-5916786-A Method for the production of chiral 1,3-aminoalcohols BIOCATALYTICS, INC. (US) 1999-06-29 US disclosed