SCHEMBL791102

SCHEMBL791102

COc1ncc(B2OC(C)(C)C(C)(C)O2)cc1NS(=O)(=O)c1cccnc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALPL P05186 1/20 0.52
PIK3CA P42336 3/20 0.51
MTOR P42345 2/20 0.51
SLC40A1 Q9NP59 6/20 0.50
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
PIK3CG P48736 3/20 0.45
PI4KA P42356 1/20 0.45
BRAF P15056 2/20 0.44
GLO1 Q04760 1/20 0.44
PIK3CD O00329 2/20 0.43
PIK3R1 P27986 1/20 0.43
PIK3CB P42338 1/20 0.43
NAMPT P43490 1/20 0.43
GAA P10253 1/20 0.42
CYP17A1 P05093 1/20 0.42
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29556249 1.00 ALPL (0.52) ALPLPIK3CAMTORSLC40A1KEAP1
SCHEMBL29556839 0.91 ALPL (0.56) ALPLPIK3CAMTORSLC40A1PIK3CG
SCHEMBL790824 0.91 ALPL (0.56) ALPLPIK3CAMTORSLC40A1PIK3CG
SCHEMBL28554047 0.90 ALPL (0.51) ALPLPIK3CAMTORSLC40A1PIK3CG
SCHEMBL798317 0.90 ALPL (0.44) ALPLPIK3CAMTORSLC40A1KEAP1
SCHEMBL15459550 0.86 ALPL (0.51) ALPLPIK3CAMTORPIK3CGPI4KA
SCHEMBL15462778 0.86 ALPL (0.51) ALPLPIK3CAMTORSLC40A1KEAP1
SCHEMBL15650005 0.85 ALPL (0.50) ALPLPIK3CAMTORPIK3CGPIK3CD
SCHEMBL15559069 0.85 ALPL (0.52) ALPLPIK3CAMTORPIK3CGBRAF
SCHEMBL22508714 0.85 ALPL (0.50) ALPLPIK3CAMTORPIK3CGPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112724134-B Azaindazole bipyridine derivative myeloid cell proliferation inhibitor, preparation method and application thereof in pharmacy 复旦大学 2022-04-01 CN disclosed
CN-112724134-A Azaindazole bipyridine derivative myeloid cell proliferation inhibitor, preparation method and application thereof in pharmacy 复旦大学 2021-04-30 CN disclosed
WO-2015120737-A1 SUBSTITUTED PYRIDOPYRIMIDINE COMPOUNDS, PREPARATION METHODS THEREFOR AND USES THEREOF 北大方正集团有限公司 2015-08-20 WO disclosed
WO-2012174312-A2 BENZIMIDAZOLE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-12-20 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed