SCHEMBL7911281

SCHEMBL7911281

COc1ccc(S(=O)(=O)NCCc2ccc(C#N)cc2)cc1

nearest known ligand 0.79

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.79
SMN1; SMN2 Q16637 2/20 0.79
POLB P06746 2/20 0.69
LSS P48449 2/20 0.65
PKM P14618 1/20 0.58
CYP19A1 P11511 1/20 0.57
SGMS1 Q86VZ5 1/20 0.56
CA12 O43570 1/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
CA5A P35218 1/20 0.56
CA9 Q16790 1/20 0.56
CA14 Q9ULX7 1/20 0.56
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
AKR1C3 P42330 1/20 0.54
MAPT P10636 1/20 0.54
PPARG P37231 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7113122 0.89 ALDH1A1 (1.00) ALDH1A1SMN1; SMN2POLBPKMSGMS1
SCHEMBL9272868 0.86 ALDH1A1 (0.65) ALDH1A1SMN1; SMN2POLBLSSSGMS1
SCHEMBL7877042 0.84 PDE4A (0.65) ALDH1A1SMN1; SMN2POLBLSSCA12
SCHEMBL15619063 0.83 ALDH1A1 (0.88) ALDH1A1SMN1; SMN2POLBPKMCA12
SCHEMBL11335294 0.83 ALDH1A1 (0.88) ALDH1A1SMN1; SMN2POLBPKMSGMS1
SCHEMBL10523408 0.82 ALDH1A1 (0.86) ALDH1A1SMN1; SMN2POLBPKMSGMS1
SCHEMBL10462588 0.82 LSS (0.67) ALDH1A1SMN1; SMN2LSSCYP19A1CA12
SCHEMBL29259796 0.82 ALDH1A1 (0.86) ALDH1A1SMN1; SMN2POLBPKMSGMS1
SCHEMBL6799293 0.82 ALDH1A1 (0.86) ALDH1A1SMN1; SMN2POLBPKMSGMS1
SCHEMBL5188475 0.82 ALDH1A1 (0.81) ALDH1A1SMN1; SMN2POLBPKMSGMS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6215001-B1 ANTIINFLAMMATORY AGENTS, ANTIASTHMATICS, AND ANTIALLERGENS; SIDE EFFECT REDUCTION KNOLL AKTIENGESELLSCHAFT (DE) 2001-04-10 US disclosed
US-6031109-A Phenoxy-, phenylthio-, benzoyl-alkyleneaminoalkylene-imidazole derivatives as therapeutic agents KNOLL AKTIENGESELLSCHAFT (DE) 2000-02-29 US disclosed
US-5780642-A NON-STEROIDAL ANTIINFLAMMATORY AGENT WHICH BLOCKS RELEASE OF ARACHIDONIC ACID FROM PHOSPHOLIPIDS; SIDE EFFECT REDUCTION KNOLL AKTIENGESELLSCHAFT (DE) 1998-07-14 US disclosed
WO-1995000493-A1 IMIDAZOLE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL AG (DE) 1995-01-05 WO disclosed