SCHEMBL7912461

SCHEMBL7912461

C[C@H](NC(=O)C1(c2ccccc2)CCN(C(=O)c2ccc(N3CCCC3=O)cc2)CC1)C1=CC=CCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
HPGD P15428 4/20 0.47
ALDH1A1 P00352 5/20 0.45
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
RAB9A P51151 2/20 0.39
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7908933 0.88 TSHR (0.41) CYP1A2CYP2C9ALDH1A1TSHRMEN1
SCHEMBL13092201 0.86 CYP1A2 (0.64) CYP1A2CYP2D6CYP2C9HPGDALDH1A1
SCHEMBL13092236 0.85 CYP1A2 (0.61) CYP1A2CYP2D6CYP2C9HPGDALDH1A1
SCHEMBL7912463 0.84 CA12 (0.37) ALDH1A1TSHRLMNARAB9ACA12
SCHEMBL7909508 0.82 CA12 (0.37) ALDH1A1TSHRMEN1KMT2ACA12
SCHEMBL7912598 0.80 CA12 (0.39) CYP1A2HPGDALDH1A1TSHRMEN1
SCHEMBL7902195 0.79 ABL1 (0.44) ALDH1A1TSHRCA12CA1CA2
SCHEMBL7910802 0.79 TSHR (0.39) ALDH1A1TSHRMEN1KMT2ASMN1; SMN2
SCHEMBL7915828 0.79 TSHR (0.39) ALDH1A1KDM4ETSHRLMNARAB9A
SCHEMBL7908120 0.79 MGLL (0.42) ALDH1A1MAPTTSHRLMNACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010106081-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-23 WO disclosed