SCHEMBL7915828

SCHEMBL7915828

C[C@H](NC(=O)C1(c2ccccc2)CCN(C(=O)c2ccc(-c3cnco3)cc2)CC1)C1=CC=CCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.39
PRLHR P49683 4/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
ALOX15 P16050 1/20 0.35
ALDH1A1 P00352 3/20 0.35
LMNA P02545 2/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.35
RAB9A P51151 1/20 0.35
GPR119 Q8TDV5 4/20 0.35
SCD5 Q86SK9 1/20 0.35
SLC9A1 P19634 1/20 0.35
HDAC4 P56524 1/20 0.34
ATM Q13315 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13092187 0.86 TSHR (0.44) TSHRPRLHRCA12CA1CA2
SCHEMBL7910802 0.86 TSHR (0.39) TSHRCA12CA1CA2CA7
SCHEMBL7908120 0.83 MGLL (0.42) TSHRCA12CA1CA2CA7
SCHEMBL7909508 0.83 CA12 (0.37) TSHRCA12CA1CA2CA7
SCHEMBL7902195 0.82 ABL1 (0.44) TSHRCA12CA1CA2CA7
SCHEMBL7912463 0.82 CA12 (0.37) TSHRCA12CA1CA2CA7
SCHEMBL7908933 0.81 TSHR (0.41) TSHRCA12CA1CA2CA7
SCHEMBL7912598 0.81 CA12 (0.39) TSHRCA12CA1CA2CA7
SCHEMBL7902201 0.81 RAB9A (0.48) TSHRCA12CA1CA2CA7
SCHEMBL7912461 0.79 CYP1A2 (0.47) TSHRCA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010106081-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-23 WO disclosed