SCHEMBL7912966

SCHEMBL7912966

COCc1nc2c(cc1C(=O)NC(=N)N)CCCCC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.43
SLC9A1 P19634 1/20 0.43
MAPT P10636 9/20 0.38
SMN1; SMN2 Q16637 7/20 0.38
ALDH1A1 P00352 7/20 0.38
RAB9A P51151 7/20 0.38
NPC1 O15118 6/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
KMT2A Q03164 2/20 0.37
PPARG P37231 1/20 0.37
NCOR2 Q9Y618 1/20 0.37
POLB P06746 6/20 0.37
TP53 P04637 5/20 0.36
USP2 O75604 1/20 0.36
HPGD P15428 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL926631 0.88 SLC9A1 (0.43) KDM4ESLC9A1MAPTSMN1; SMN2ALDH1A1
SCHEMBL7913104 0.87 KDM4E (0.45) KDM4ESLC9A1MAPTSMN1; SMN2ALDH1A1
SCHEMBL927564 0.86 KDM4E (0.38) KDM4ESLC9A1MAPTSMN1; SMN2ALDH1A1
SCHEMBL7913003 0.85 SLC9A1 (0.43) KDM4ESLC9A1MAPTSMN1; SMN2ALDH1A1
SCHEMBL7911317 0.84 SLC9A1 (0.43) KDM4ESLC9A1MAPTSMN1; SMN2ALDH1A1
SCHEMBL927565 0.84 KDM4E (0.37) KDM4ESLC9A1MAPTSMN1; SMN2ALDH1A1
SCHEMBL7916722 0.82 SLC9A1 (0.45) KDM4ESLC9A1MAPTSMN1; SMN2ALDH1A1
SCHEMBL7913282 0.82 KDM4E (0.49) KDM4ESLC9A1MAPTSMN1; SMN2ALDH1A1
SCHEMBL7916794 0.81 SLC9A1 (0.61) KDM4ESLC9A1MAPTSMN1; SMN2ALDH1A1
SCHEMBL927184 0.81 SLC9A1 (0.61) KDM4ESLC9A1MAPTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6258829-B1 ANTIARRTHMIA AGENTS AND CARDIOVASCULAR DISORDERS TOA EIYO LTD. (JP) 2001-07-10 US disclosed
EP-0972767-A1 CYCLOALKA[b]PYRIDINE-3-CARBONYLGUANIDINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, AND DRUGS CONTAINING THE SAME TOA EIYO LTD. (JP) 2000-01-19 EP disclosed