SCHEMBL7913073

SCHEMBL7913073

Nc1c(Nc2cccc(-c3cc4ccccc4[nH]3)c2)c(=O)c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.48
RAB9A P51151 4/20 0.48
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
POLB P06746 1/20 0.46
KDR P35968 2/20 0.46
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
VCP P55072 2/20 0.41
SMO Q99835 1/20 0.41
CYP19A1 P11511 1/20 0.41
KDM4E B2RXH2 3/20 0.40
MAPT P10636 3/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
CASP3 P42574 2/20 0.40
SENP8 Q96LD8 2/20 0.40
SENP7 Q9BQF6 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7913077 0.78 KDM4E (0.57) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL7905830 0.78 SIRT2 (0.48) MEN1KMT2APOLBCA2CA9
SCHEMBL7905887 0.75 APP (0.50) CA12CA1CA2CA9TBK1
SCHEMBL14303521 0.74 NPC1 (0.61) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL8304969 0.72 NPC1 (0.80) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL11724742 0.72 NPC1 (0.67) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL7914160 0.71 CXCR2 (0.43) MEN1KMT2APOLBKDRALDH1A1
SCHEMBL6925698 0.70 NPC1 (0.56) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL7913081 0.70 HDAC3 (0.46) MEN1KMT2APOLBCYP2C9
SCHEMBL7916081 0.70 CNR1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211220-B1 ANTITUMOR AGENTS AND ANTICARCIINOGENIC AGENTS CELL PATHWAYS, INC. 2001-04-03 US claimed
US-6211220-B1 ANTITUMOR AGENTS AND ANTICARCIINOGENIC AGENTS CELL PATHWAYS, INC. 2001-04-03 US disclosed
WO-1994029277-A1 AMILINO- OR PYRIDYLAMINO- CYCLOBUTENE- 1,2-DIONE DERIVATIVES AS cGMP PHOSPHODIESTERASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1994-12-22 WO disclosed