SCHEMBL7913110

SCHEMBL7913110

Cc1cc2c(=O)[nH]nc(-c3ccccc3)n2n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
PARP1 P09874 2/20 0.44
CYP1A2 P05177 1/20 0.44
ATM Q13315 2/20 0.43
NPSR1 Q6W5P4 1/20 0.39
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
TYK2 P29597 1/20 0.38
JAK3 P52333 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.38
HSD17B10 Q99714 3/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38
POLB P06746 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5710845 0.78 NPC1 (0.51) NPC1RAB9APARP1CYP1A2MEN1
SCHEMBL31309174 0.74 PARP1 (0.39) NPC1RAB9APARP1CYP1A2ATM
SCHEMBL23950159 0.72 PARP1 (0.37) NPC1RAB9APARP1CYP1A2ATM
SCHEMBL30273093 0.69 PARP1 (0.54) NPC1RAB9APARP1CYP1A2KMT2A
SCHEMBL8480564 0.67 JAK2 (0.51) ATMNPSR1JAK2JAK1TYK2
SCHEMBL21851805 0.67 ALDH1A1 (0.39) NPC1RAB9ANPSR1MEN1KMT2A
SCHEMBL4871941 0.66 CYP1A2 (0.41) NPC1RAB9APARP1CYP1A2MEN1
SCHEMBL3520851 0.66 PDE3B (0.47) KMT2AKDM4EALDH1A1HSD17B10HPGD
SCHEMBL16506739 0.66 PARP1 (0.68) NPC1RAB9APARP1CYP1A2ADORA3
SCHEMBL18752187 0.66 AKT2 (0.44) NPC1RAB9ANPSR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed