SCHEMBL7913459

SCHEMBL7913459

COc1ccc(C(=O)c2ccccc2)cc1OC1Cc2ccccc2C1

nearest known ligand 0.70

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 8/20 0.70
PDE4A P27815 7/20 0.70
PDE4B Q07343 7/20 0.70
PDE4C Q08493 7/20 0.70
CYP1A2 P05177 2/20 0.55
CYP2C19 P33261 2/20 0.55
CYP2D6 P10635 1/20 0.55
HPGD P15428 1/20 0.55
CYP3A4 P08684 1/20 0.54
CYP2C9 P11712 1/20 0.54
TSHR P16473 1/20 0.54
PDE5A O76074 1/20 0.54
ACHE P22303 3/20 0.53
BCHE P06276 2/20 0.53
ALDH1A1 P00352 1/20 0.51
GAA P10253 1/20 0.51
PTGS1 P23219 1/20 0.50
PTGS2 P35354 1/20 0.50
NOX1 Q9Y5S8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3371531 0.86 PDE4D (0.69) PDE4DPDE4APDE4BPDE4CPDE5A
SCHEMBL4162765 0.85 PDE5A (0.70) PDE4DPDE4APDE4BPDE4CPDE5A
SCHEMBL7441489 0.82 PDE4B (0.63) PDE4DPDE4APDE4BPDE4C
SCHEMBL1333620 0.81 CYP1A2 (0.81) CYP1A2CYP2C19CYP2D6HPGDCYP3A4
SCHEMBL4825206 0.80 PDE4B (0.61) PDE4DPDE4APDE4BPDE4CALDH1A1
SCHEMBL7366699 0.79 PDE4B (0.62) PDE4DPDE4APDE4BPDE4CALDH1A1
SCHEMBL9184286 0.79 PDE4B (0.62) PDE4DPDE4APDE4BPDE4CALDH1A1
SCHEMBL7359869 0.78 MAPT (0.67) PDE4DPDE4APDE4BPDE4CHPGD
SCHEMBL27472680 0.77 PDE4D (0.68) PDE4DPDE4APDE4BPDE4CCYP1A2
SCHEMBL3371565 0.77 PDE4B (0.57) PDE4DPDE4APDE4BPDE4CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265402-B1 ANTIINFLAMMATORY AGENTS NIKKEN CHEMICALS CO., LTD. (JP) 2001-07-24 US disclosed
EP-0924204-A1 2-PHENYLMORPHOLIN-5-ONE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME Nikken Chemicals Company, Limited (JP) 1999-06-23 EP disclosed