SCHEMBL7913593

SCHEMBL7913593

O=c1cc(-c2ccc3ccccc3c2)[nH]c2ncccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.72
ADORA1 P30542 5/20 0.72
RIPK1 Q13546 3/20 0.54
KDM4E B2RXH2 1/20 0.47
GMNN O75496 1/20 0.47
LMNA P02545 1/20 0.47
CYP1A2 P05177 1/20 0.47
PKM P14618 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
MTOR P42345 1/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
HIF1A Q16665 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CCNB2 O95067 1/20 0.47
CDK1 P06493 1/20 0.47
CCNB1 P14635 1/20 0.47
CCNB3 Q8WWL7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3866419 0.84 ADORA2A (1.00) ADORA2AADORA1KDM4EGMNNLMNA
SCHEMBL7913586 0.80
SCHEMBL7921812 0.80 KDM4E (0.47) ADORA2AADORA1KDM4EGMNNLMNA
SCHEMBL7921814 0.80 ADORA2A (0.76) ADORA2AADORA1LMNACCNB2CDK1
SCHEMBL7925170 0.80 ADORA2A (0.76) ADORA2AADORA1KDM4EGMNNLMNA
SCHEMBL30472919 0.80 ADORA2A (0.70) ADORA2AADORA1RIPK1KDM4ELMNA
SCHEMBL7920130 0.80 ADORA2A (0.75) ADORA2AADORA1
SCHEMBL7913613 0.80 ADORA2A (0.70) ADORA2AADORA1RIPK1KDM4ELMNA
SCHEMBL7925077 0.79 ADORA2A (0.65) ADORA2AADORA1RIPK1KDM4E
SCHEMBL31238215 0.79 ADORA2A (0.65) ADORA2AADORA1RIPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6229016-B1 PYRIDOPYRIMIDINE DERIVATIVES AS CHEMICAL INTERMEDIATES; POLYMERIZATION INHIBITION OF TUBULIN THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL 2001-05-08 US disclosed
US-6071930-A FOR INHIBITION OF MITOSIS OR TUMOR GROWTH THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2000-06-06 US disclosed
EP-0971921-A1 2-ARYL-NAPHTHYRIDIN-4-ONES AS ANTITUMOR AGENTS The University of North Carolina at Chapel Hill (US) 2000-01-19 EP disclosed
US-5994367-A PREVENT CELL MITOSIS; ANTICARCINOGENIC AGENTS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1999-11-30 US disclosed
WO-1998039332-A1 2-ARYL-NAPHTHYRIDIN-4-ONES AS ANTITUMOR AGENTS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1998-09-11 WO disclosed