SCHEMBL7925170

SCHEMBL7925170

O=c1cc(-c2ccc(Cl)cc2)[nH]c2ncccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.76
ADORA1 P30542 2/20 0.76
KDM4E B2RXH2 2/20 0.60
PDE10A Q9Y233 2/20 0.60
KMT2A Q03164 2/20 0.60
CCNB2 O95067 1/20 0.55
CDK1 P06493 1/20 0.55
CCNB1 P14635 1/20 0.55
CCNB3 Q8WWL7 1/20 0.55
GMNN O75496 1/20 0.52
LMNA P02545 1/20 0.52
CYP1A2 P05177 1/20 0.52
PKM P14618 1/20 0.52
TSHR P16473 1/20 0.52
CYP2C19 P33261 1/20 0.52
MTOR P42345 1/20 0.52
BLM P54132 1/20 0.52
PMP22 Q01453 1/20 0.52
HIF1A Q16665 1/20 0.52
HSD17B10 Q99714 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3866419 0.86 ADORA2A (1.00) ADORA2AADORA1KDM4ECCNB2CDK1
SCHEMBL31061064 0.86 ADORA2A (0.72) ADORA2AADORA1KDM4EGMNNLMNA
SCHEMBL7920166 0.86 ADORA2A (0.72) ADORA2AADORA1KDM4EGMNNLMNA
SCHEMBL7921814 0.85 ADORA2A (0.76) ADORA2AADORA1CCNB2CDK1CCNB1
SCHEMBL27167216 0.82 ADORA2A (0.70) ADORA2AADORA1
SCHEMBL12424812 0.82 ADORA2A (0.58) ADORA2AADORA1KMT2AMEN1ALDH1A1
SCHEMBL7913613 0.82 ADORA2A (0.70) ADORA2AADORA1KDM4EKMT2ACCNB2
SCHEMBL30472919 0.82 ADORA2A (0.70) ADORA2AADORA1KDM4EKMT2ACCNB2
SCHEMBL7913593 0.80 ADORA2A (0.72) ADORA2AADORA1KDM4ECCNB2CDK1
SCHEMBL31265224 0.78 RIPK1 (0.71) CCNB2CDK1CCNB1CCNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6229016-B1 PYRIDOPYRIMIDINE DERIVATIVES AS CHEMICAL INTERMEDIATES; POLYMERIZATION INHIBITION OF TUBULIN THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL 2001-05-08 US disclosed
US-6071930-A FOR INHIBITION OF MITOSIS OR TUMOR GROWTH THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2000-06-06 US disclosed
EP-0971921-A1 2-ARYL-NAPHTHYRIDIN-4-ONES AS ANTITUMOR AGENTS The University of North Carolina at Chapel Hill (US) 2000-01-19 EP disclosed
US-5994367-A PREVENT CELL MITOSIS; ANTICARCINOGENIC AGENTS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1999-11-30 US disclosed
WO-1998039332-A1 2-ARYL-NAPHTHYRIDIN-4-ONES AS ANTITUMOR AGENTS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1998-09-11 WO disclosed