SCHEMBL7916623

SCHEMBL7916623

FC(F)(F)c1cnc(OCc2ccccc2)c(Br)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 2/20 0.51
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
LRRK2 Q5S007 2/20 0.41
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
SLC6A4 P31645 2/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
MAOB P27338 2/20 0.40
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SLC6A9 P48067 1/20 0.39
HPGD P15428 1/20 0.39
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30104807 1.00 MRGPRX4 (0.51) MRGPRX4ALDH1A1MEN1KMT2ALRRK2
SCHEMBL4284174 0.84 MRGPRX4 (0.52) MRGPRX4ALDH1A1MEN1KMT2ALRRK2
SCHEMBL4160021 0.84 MRGPRX4 (0.52) MRGPRX4ALDH1A1MEN1KMT2ALRRK2
SCHEMBL8431628 0.84 MRGPRX4 (0.52) MRGPRX4ALDH1A1MEN1KMT2ALRRK2
SCHEMBL6743790 0.82 MRGPRX4 (0.71) MRGPRX4ALDH1A1MEN1KMT2ACYP1A2
SCHEMBL31730574 0.80 MAOB (0.42) ALDH1A1LRRK2THRATHRBSLC6A4
SCHEMBL1542659 0.80 MAOB (0.42) ALDH1A1LRRK2THRATHRBSLC6A4
SCHEMBL17594985 0.80 MAOB (0.49) ALDH1A1THRATHRBSLC6A4MAOB
SCHEMBL31730474 0.79 MRGPRX4 (0.51) MRGPRX4ALDH1A1MEN1KMT2ALRRK2
SCHEMBL4146898 0.79 MRGPRX4 (0.51) MRGPRX4ALDH1A1MEN1KMT2ALRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396485-A PARP7 inhibitors 轩竹生物科技股份有限公司 2024-01-12 CN disclosed
US-6225320-B1 TREATMENT OF PAIN, INFLAMMATION, MIGRAINE, EMESIS AND POSTTHERPETIC NEURALGIA MERCK SHARP & DOHME LTD. (GB) 2001-05-01 US disclosed
EP-0989987-A1 SPIRO-AZACYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 2000-04-05 EP disclosed
WO-1998054187-A1 SPIRO-AZACYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 1998-12-03 WO disclosed