SCHEMBL7917480

SCHEMBL7917480

COCCOc1ncc(C(F)(F)F)cc1Br

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HTT P42858 2/20 0.36
KDM4E B2RXH2 1/20 0.36
KMT2A Q03164 1/20 0.36
APP P05067 5/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
PTGS2 P35354 1/20 0.36
PPARG P37231 4/20 0.36
MALT1 Q9UDY8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7909812 0.86 ALDH1A1 (0.37) LMNAALDH1A1HPGDKMT2AAPP
SCHEMBL18600965 0.83 APP (0.50) ALDH1A1SMN1; SMN2HTTAPPPTGS2
SCHEMBL6502269 0.82 NPSR1 (0.44) LMNAALDH1A1HPGDKMT2ACYP1A2
SCHEMBL29837917 0.82 CYP1A2 (0.43) LMNAHPGDSMN1; SMN2KDM4EKMT2A
SCHEMBL7916612 0.82 CYP1A2 (0.43) LMNAHPGDSMN1; SMN2KDM4EKMT2A
SCHEMBL22278620 0.81 APP (0.33) HPGDKMT2AAPPCYP1A2CYP3A4
SCHEMBL15716504 0.81 CYP1A2 (0.45) LMNAALDH1A1HPGDSMN1; SMN2HTT
SCHEMBL7917315 0.80 PTGS2 (0.48) ALDH1A1HPGDSMN1; SMN2KDM4EKMT2A
SCHEMBL22638138 0.76 SSTR4 (0.44) ALDH1A1HPGDSMN1; SMN2HTTKDM4E
SCHEMBL29749337 0.76 SSTR4 (0.44) ALDH1A1HPGDSMN1; SMN2HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6225320-B1 TREATMENT OF PAIN, INFLAMMATION, MIGRAINE, EMESIS AND POSTTHERPETIC NEURALGIA MERCK SHARP & DOHME LTD. (GB) 2001-05-01 US disclosed
EP-0989987-A1 SPIRO-AZACYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 2000-04-05 EP disclosed
WO-1998054187-A1 SPIRO-AZACYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 1998-12-03 WO disclosed