SCHEMBL7918503

SCHEMBL7918503

C[C@H](CC1CCC1)NC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(Oc2ccccc2)nc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRN P28799 2/20 0.53
SORT1 Q99523 2/20 0.53
OPRM1 P35372 1/20 0.51
OPRD1 P41143 1/20 0.51
CTSA P10619 2/20 0.49
ACACB O00763 4/20 0.47
PSMB11 A5LHX3 1/20 0.46
PSMA7 O14818 1/20 0.46
PSMB1 P20618 1/20 0.46
PSMA1 P25786 1/20 0.46
PSMA2 P25787 1/20 0.46
PSMA3 P25788 1/20 0.46
PSMA4 P25789 1/20 0.46
PSMB8 P28062 1/20 0.46
PSMB9 P28065 1/20 0.46
PSMA5 P28066 1/20 0.46
PSMB4 P28070 1/20 0.46
PSMB6 P28072 1/20 0.46
PSMB5 P28074 1/20 0.46
LONP1 P36776 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3148974 0.88 PSMB5 (0.61) GRNSORT1OPRM1OPRD1CTSA
SCHEMBL19381926 0.88 PSMB5 (0.61) GRNSORT1OPRM1OPRD1CTSA
SCHEMBL7921841 0.73 IKBKB (0.41) PSMB11PSMA7PSMB1PSMA1PSMA2
SCHEMBL19382404 0.73 PSMB5 (0.53) ACACBPSMB11PSMA7PSMB1PSMA1
SCHEMBL3143565 0.73 PSMB5 (0.53) ACACBPSMB11PSMA7PSMB1PSMA1
SCHEMBL19382408 0.71 CTSS (0.51) GPR139CTSS
SCHEMBL3144997 0.71 PSMB5 (0.57) PSMB11PSMA7PSMB1PSMA1PSMA2
SCHEMBL19381925 0.71 USP30 (0.46) CTSS
SCHEMBL24283548 0.70 GRN (1.00) GRNSORT1OPRM1OPRD1CTSA
SCHEMBL24283501 0.69 GRN (0.78) GRNSORT1OPRM1OPRD1CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036357-A1 DERIVATIVES OF 1-AMINO-2-CYCLOBUTYLETHYLBORONIC ACID MILLENNIUM PHARMACEUTICALS, INC. (US) 2010-04-01 WO disclosed