SCHEMBL7918903

SCHEMBL7918903

CCCCn1c(=O)c2[nH]c(C)nc2n(CCCC)c1=O

nearest known ligand 0.82

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.57
ADORA2A P29274 2/20 0.57
ADORA3 P0DMS8 1/20 0.57
ADORA2B P29275 1/20 0.57
SIRT1 Q96EB6 1/20 0.56
SIRT3 Q9NTG7 1/20 0.56
SIRT5 Q9NXA8 1/20 0.56
PDE2A O00408 1/20 0.54
PDE1A P54750 1/20 0.54
PDE1B Q01064 1/20 0.54
PDE1C Q14123 1/20 0.54
PDE4A P27815 1/20 0.54
PDE4B Q07343 1/20 0.54
PDE4C Q08493 1/20 0.54
PDE4D Q08499 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10859893 0.97 SIRT1 (0.61) ADORA1ADORA2ASIRT1SIRT3SIRT5
SCHEMBL10856971 0.97 SIRT1 (0.61) ADORA1ADORA2ASIRT1SIRT3SIRT5
SCHEMBL11072524 0.94 SIRT1 (0.55) ADORA1ADORA2AADORA3ADORA2BSIRT1
SCHEMBL1063544 0.90 SIRT1 (0.68) ADORA1ADORA2AADORA3ADORA2BSIRT1
SCHEMBL11066305 0.90 SIRT1 (0.54) ADORA1ADORA2AADORA3ADORA2BSIRT1
SCHEMBL10855008 0.89 ADORA2A (0.49) ADORA1ADORA2AADORA3ADORA2BSIRT1
SCHEMBL4953015 0.88 ADORA2B (0.52) ADORA1ADORA2AADORA3ADORA2BSIRT1
SCHEMBL10861347 0.87 PDE2A (0.54) ADORA1ADORA2AADORA3ADORA2BSIRT1
SCHEMBL9430619 0.87 ADORA2A (0.61) ADORA1ADORA2AADORA3ADORA2BSIRT1
SCHEMBL1462066 0.86 PDE2A (0.46) ADORA1ADORA2AADORA3ADORA2BSIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6221874-B1 7-CYCLIC-SUBSTITUTED SULFONYL-3,7-DIHYDRO-PURINE-2, 6-DIONE DERIVATIVES AMERICAN HOME PRODUCTS CORPORATION 2001-04-24 US disclosed
EP-0708781-A1 A 3 ADENOSINE RECEPTOR AGONISTS THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, Department of Health and Human Services (US) 1996-05-01 EP disclosed