SCHEMBL7920280

SCHEMBL7920280

COc1ccc(-c2cc(C(F)(F)F)nn2-c2ccccc2S(N)(=O)=O)cc1F

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.58
PTGS1 P23219 8/20 0.56
ABCB11 O95342 1/20 0.51
ALDH1A1 P00352 1/20 0.51
PDPK1 O15530 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8692194 0.93 PTGS2 (0.50) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8689608 0.92 PTGS2 (0.49) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8639264 0.92 PTGS2 (0.69) PTGS2PTGS1PDPK1
SCHEMBL8639247 0.90 PTGS2 (0.70) PTGS2PTGS1ABCB11PDPK1
SCHEMBL8689327 0.89 PTGS2 (0.57) PTGS2PTGS1PDPK1
SCHEMBL8525531 0.89 PTGS2 (0.48) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL8694131 0.88 PTGS2 (0.71) PTGS2PTGS1PDPK1
SCHEMBL8689089 0.88 PTGS2 (0.56) PTGS2PTGS1PDPK1
SCHEMBL8693509 0.86 PTGS2 (0.62) PTGS2PTGS1PDPK1
SCHEMBL8688624 0.86 PTGS2 (0.54) PTGS2PTGS1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2001527542-A 2001-12-25 JP claimed
EP-0979077-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE PREVENTION OF CARDIOVASCULAR DISORDERS G.D. Searle & Co. (US) 2000-02-16 EP claimed
WO-1998047509-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE PREVENTION OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1998-10-29 WO claimed
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US claimed
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5753688-A ANTIINFLAMMATORY TALLEY JOHN J (US) 1998-05-19 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed