SCHEMBL8525531

SCHEMBL8525531

COc1ccc(-c2cc(C(F)(F)F)nn2-c2ccccc2S(N)(=O)=O)cc1F.NS(=O)(=O)c1ccccc1-n1ncc(Cl)c1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.48
PTGS1 P23219 9/20 0.47
RXRA P19793 2/20 0.45
NR1H2 P55055 2/20 0.45
NR1H3 Q13133 2/20 0.45
PDPK1 O15530 1/20 0.43
ABCB11 O95342 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7920280 0.89 PTGS2 (0.58) PTGS2PTGS1PDPK1ABCB11ALDH1A1
SCHEMBL8689327 0.85 PTGS2 (0.57) PTGS2PTGS1RXRANR1H2NR1H3
SCHEMBL8689608 0.84 PTGS2 (0.49) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8692194 0.83 PTGS2 (0.50) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8639264 0.82 PTGS2 (0.69) PTGS2PTGS1RXRANR1H2NR1H3
SCHEMBL8639247 0.80 PTGS2 (0.70) PTGS2PTGS1PDPK1ABCB11
SCHEMBL8688677 0.79 PTGS2 (0.56) PTGS2PTGS1RXRANR1H2NR1H3
SCHEMBL8694131 0.79 PTGS2 (0.71) PTGS2PTGS1PDPK1
SCHEMBL8689089 0.78 PTGS2 (0.56) PTGS2PTGS1PDPK1
SCHEMBL8691904 0.78 PTGS2 (0.49) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998016227-A9 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE TREATMENT AND PREVENTION OF NEOPLASIA 1998-07-30 WO claimed
EP-0941080-A2 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS AS ANTI-ANGIOGENIC AGENTS G.D. SEARLE & CO. (US) 1999-09-15 EP disclosed
WO-1998022101-A2 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS AS ANTI-ANGIOGENIC AGENTS G.D. SEARLE & CO. (US) 1998-05-28 WO disclosed