SCHEMBL7921100

SCHEMBL7921100

CC1C(CN2CCCC2)N(C(=O)Cc2ccc(Cl)c(Cl)c2)CCN1C(=O)O

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 16/20 0.68
UTS2R Q9UKP6 1/20 0.64
OPRD1 P41143 3/20 0.61
CYP3A4 P08684 2/20 0.61
CYP2D6 P10635 2/20 0.61
CYP2C9 P11712 2/20 0.61
CYP2C19 P33261 2/20 0.61
TDP1 Q9NUW8 2/20 0.61
NPC1 O15118 1/20 0.61
CYP1A2 P05177 1/20 0.61
NFKB1 P19838 1/20 0.61
HIF1A Q16665 1/20 0.61
BLM P54132 1/20 0.60
PMP22 Q01453 1/20 0.60
DRD4 P21917 1/20 0.60
SLC6A3 Q01959 1/20 0.60
TMEM97 Q5BJF2 1/20 0.60
SIGMAR1 Q99720 1/20 0.60
OPRM1 P35372 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8819811 0.95 OPRK1 (0.62) OPRK1UTS2ROPRD1CYP3A4CYP2D6
Fumaric Acid SCHEMBL7947009 0.95 OPRK1 (0.62) OPRK1UTS2ROPRD1CYP3A4CYP2D6
Fumaric Acid SCHEMBL7647035 0.95 OPRK1 (0.62) OPRK1UTS2ROPRD1CYP3A4CYP2D6
SCHEMBL9515474 0.83 OPRK1 (0.80) OPRK1UTS2ROPRD1CYP3A4CYP2D6
Fumaric Acid SCHEMBL10417793 0.83 HPGD (0.51) OPRK1UTS2ROPRD1CYP3A4CYP2D6
SCHEMBL9514408 0.81 OPRK1 (1.00) OPRK1UTS2ROPRD1CYP3A4CYP2D6
Fumaric Acid SCHEMBL9734432 0.81 OPRK1 (0.71) OPRK1UTS2ROPRD1CYP3A4CYP2D6
Maleic Acid SCHEMBL9734427 0.81 OPRK1 (0.71) OPRK1UTS2ROPRD1CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9734739 0.80 OPRK1 (0.98) OPRK1UTS2ROPRD1CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9733562 0.80 OPRK1 (0.98) OPRK1UTS2ROPRD1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174891-B1 A MORPHINAN DERIVTIVE AS A POTENT AND FAST-ACTING OPIATE KAPPA RECEPTOR FOR THE RELIEF OF PURITIS DUE TO DERMATOSES WITH INFLAMMATION OR AN INTERNAL DISEASE (MALIGNANT TUMORS, DIABETES MELLITUS, HEPATIC DISEASES, GOUT; RENAL FAILURE TORAY INDUSTRIES, INC. (JP) 2001-01-16 US disclosed