SCHEMBL7921968

SCHEMBL7921968

COC(=O)Nc1ccc2c(c1)CC1(COC(N)=N1)C2

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
BACE1 P56817 16/20 0.39
BACE2 Q9Y5Z0 10/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7917963 0.91 BACE1 (0.43) MEN1KMT2ABACE1BACE2KCNH2
SCHEMBL7918038 0.91 BACE1 (0.43) MEN1KMT2ABACE1BACE2KCNH2
SCHEMBL7924845 0.88 CYP1A2 (0.42) BACE1BACE2
SCHEMBL7913188 0.86 BACE1 (0.39) KMT2ABACE1BACE2KCNH2
SCHEMBL7920108 0.79 BACE1 (0.45) BACE1BACE2KCNH2
SCHEMBL7921890 0.77 BACE1 (0.33) BACE1BACE2KCNH2
SCHEMBL7920091 0.76 CYP1A2 (0.49) BACE1KCNH2
SCHEMBL7918102 0.74 HTT (0.34) BACE1BACE2KCNH2
SCHEMBL7918363 0.73 TAAR1 (0.51) MEN1KMT2ABACE1
SCHEMBL7919840 0.73 TAAR1 (0.51) MEN1KMT2ABACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010042475-A1 SPIROAMINOOXAZOLINE ANALOGUES AS ALPHA2C ADRENERGIC RECEPTOR MODULATORS SCHERING CORPORATION (US) 2010-04-15 WO disclosed