SCHEMBL7918038

SCHEMBL7918038

COC(=O)Nc1ccc2c(c1)CC1(CC2)COC(N)=N1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 13/20 0.43
TAAR1 Q96RJ0 1/20 0.43
ADRA2A P08913 1/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KCNH2 Q12809 2/20 0.39
BACE2 Q9Y5Z0 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7917963 0.96 BACE1 (0.43) BACE1TAAR1ADRA2AMEN1KMT2A
SCHEMBL7921968 0.91 MEN1 (0.42) BACE1MEN1KMT2AKCNH2BACE2
SCHEMBL7920108 0.84 BACE1 (0.45) BACE1TAAR1ADRA2AKCNH2BACE2
SCHEMBL7924845 0.79 CYP1A2 (0.42) BACE1ADRA2ABACE2
SCHEMBL7918363 0.78 TAAR1 (0.51) BACE1TAAR1ADRA2AMEN1KMT2A
SCHEMBL7918614 0.78 TAAR1 (0.51) BACE1TAAR1ADRA2AMEN1KMT2A
SCHEMBL7919840 0.78 TAAR1 (0.51) BACE1TAAR1ADRA2AMEN1KMT2A
SCHEMBL7918622 0.78 ADRA2A (0.60) BACE1TAAR1ADRA2AMEN1KMT2A
SCHEMBL7913188 0.77 BACE1 (0.39) BACE1KMT2AKCNH2BACE2
SCHEMBL7913281 0.76 TAAR1 (0.40) BACE1TAAR1ADRA2AKCNH2BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010042475-A1 SPIROAMINOOXAZOLINE ANALOGUES AS ALPHA2C ADRENERGIC RECEPTOR MODULATORS SCHERING CORPORATION (US) 2010-04-15 WO disclosed