SCHEMBL7922185

SCHEMBL7922185

C=CCOc1ccc(NC(C)=O)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.68
MAPT P10636 6/20 0.65
RAB9A P51151 3/20 0.65
NPC1 O15118 1/20 0.65
POLB P06746 1/20 0.65
SMN1; SMN2 Q16637 1/20 0.65
KMT2A Q03164 4/20 0.65
MEN1 O00255 3/20 0.65
CYP1A2 P05177 2/20 0.65
LMNA P02545 1/20 0.65
TDP1 Q9NUW8 1/20 0.65
ALDH1A1 P00352 4/20 0.59
KDM4E B2RXH2 1/20 0.54
HPGD P15428 1/20 0.54
HSD17B10 Q99714 1/20 0.52
GAA P10253 1/20 0.52
ADRB2 P07550 1/20 0.50
ADRB1 P08588 1/20 0.50
ADRB3 P13945 1/20 0.50
OPRK1 P41145 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22619559 0.86 MAPT (0.64) HTTMAPTRAB9ANPC1POLB
SCHEMBL9570572 0.86 HTT (0.71) HTTMAPTRAB9APOLBSMN1; SMN2
SCHEMBL9570664 0.86 HTT (0.71) HTTMAPTRAB9APOLBSMN1; SMN2
SCHEMBL7356605 0.85 HTT (0.69) HTTMAPTRAB9ASMN1; SMN2KMT2A
SCHEMBL13652531 0.84 MAPT (0.66) HTTMAPTRAB9ANPC1POLB
SCHEMBL28527575 0.83 ALDH1A1 (0.63) HTTMAPTRAB9ANPC1POLB
SCHEMBL11684715 0.83 MAPT (0.60) HTTMAPTRAB9ANPC1POLB
SCHEMBL22192215 0.82 NPC1 (0.86) MAPTRAB9ANPC1POLBSMN1; SMN2
SCHEMBL4980566 0.81 GAA (0.64) HTTMAPTRAB9ANPC1POLB
SCHEMBL1064813 0.81 KMT2A (0.71) HTTMAPTRAB9ASMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-6293719-A None JP disclosed
EP-4398037-A1 COMPOUND FOR FORMING METAL-CONTAINING FILM, COMPOSITION FOR FORMING METAL-CONTAINING FILM, AND PATTERNING PROCESS SHIN-ETSU CHEMICAL CO., LTD. (JP) 2024-07-10 EP disclosed
US-11833162-B2 Macrocyclic derivatives, process for preparing same and pharmaceutical compositions containing same LES LABORATOIRES SERVIER (FR) 2023-12-05 US disclosed
EP-3700911-B1 NOVEL MACROCYCLIC DERIVATIVES, PROCESS FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SERVIER LAB (FR) 2023-09-06 EP disclosed
CN-111511750-B Macrocyclic derivatives, process for their preparation and pharmaceutical compositions containing them 法国施维雅药厂 2023-06-13 CN disclosed
EP-3700911-A1 NOVEL MACROCYCLIC DERIVATIVES, PROCESS FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME Les Laboratoires Servier SAS (FR) 2020-09-02 EP disclosed
US-20200253993-A1 NOVEL MACROCYCLIC DERIVATIVES, PROCESS FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME LES LABORATOIRES SERVIER (FR) 2020-08-13 US disclosed
CN-111511750-A Novel macrocyclic derivatives, process for their preparation and pharmaceutical compositions containing them 法国施维雅药厂 2020-08-07 CN disclosed
WO-2019053617-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-03-21 WO disclosed
US-7576034-B2 Crosslinked three-dimensional polymer network, method for preparing same, support material comprising same and uses thereof EKA CHEMICALS AB (SE) 2009-08-18 US disclosed
EP-0934266-A1 CROSS-LINKERS FOR CROSS-LINKABLE OPTICAL POLYCARBONATES Akzo Nobel N.V. (NL) 1999-08-11 EP disclosed
US-5866611-A PHENOXYPROPYLAMINE INHIBITORS OF SQUALENE SYNTHESE, USEFUL IN TREATING DISEASES IN WHICH A LOWERING OF CHOLESTEROL IS DESIRABLE. ZENECA LIMITED (GB) 1999-02-02 US disclosed
WO-1998017644-A1 CROSS-LINKERS FOR CROSS-LINKABLE OPTICAL POLYCARBONATES AKZO NOBEL N.V. (NL) 1998-04-30 WO disclosed
JP-H06293719-A PRODUCTION OF PRIMARY AMINE HAVING THERMOSETTING GROUP KANEGAFUCHI CHEM IND CO LTD 1994-10-21 JP disclosed
EP-0589018-A1 AMINES AS INHIBITORS OF SQUALENE SYNTHASE ZENECA LIMITED (GB) 1994-03-30 EP disclosed
WO-1993020807-A1 AMINES AS INHIBITORS OF SQUALENE SYNTHASE ZENECA LIMITED (GB) 1993-10-28 WO disclosed
EP-0257391-A2 5-Substituted-3-phenyl-3-(1H-imidazol-1-ylmethyl)-2-methylisoxazolidines FISONS CORPORATION (US) 1988-03-02 EP disclosed
EP-0257351-A2 3-Phenyl-3-(1H-1,2,4-triazol-1-ylmethyl)-5-substituted-2-methyl-isoxazolidines FISONS CORPORATION (a Massachusetts corporation) (US) 1988-03-02 EP disclosed
US-4727157-A 3-(Substituted phenyl)-3-(1H-1,2,4-triazol-1-yl)methyl-2-methyl-5-[(substituted phenoxy)methyl]isoxazolidine derivatives PENNWALT CORPORATION (US) 1988-02-23 US disclosed
US-4723021-A Substituted 5-(phenoxyalkyl)-3-phenyl-3-(1H-imidazol-1-ylmethyl)-2-methylisoxazolidines PENNWALT CORPORATION (US) 1988-02-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11833162-B2 Macrocyclic derivatives, process for preparing same and pharmaceutical compositions containing same C1R, F12, RDX HTT 1693/4885MAPT 3294/4885RAB9A 1230/4885
US-20200253993-A1 NOVEL MACROCYCLIC DERIVATIVES, PROCESS FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME C1R, RDX, F12 HTT 2528/4885MAPT 3590/4885RAB9A 1298/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.