SCHEMBL7922225

SCHEMBL7922225

Cc1nc(C2(C(=O)O)C=CC(c3ccccc3C)=CC2)no1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.39
NPSR1 Q6W5P4 2/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
PKM P14618 3/20 0.34
GAA P10253 3/20 0.34
ALDH1A1 P00352 1/20 0.34
NPC1 O15118 5/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
MAPT P10636 3/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TP53 P04637 2/20 0.34
AKR1B1 P15121 1/20 0.33
RAB9A P51151 4/20 0.33
RXFP1 Q9HBX9 1/20 0.33
CASP3 P42574 1/20 0.33
SENP8 Q96LD8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28131668 0.74 MCL1 (0.37) NR1H4TP53
SCHEMBL7913508 0.71 ADORA2A (0.38) NPSR1GAAALDH1A1SMN1; SMN2MAPT
SCHEMBL27494152 0.71 NOTUM (0.45) LMNATSHRALDH1A1SMN1; SMN2MAPT
SCHEMBL28983710 0.68 GRIA1 (0.35) TSHRNPC1SMN1; SMN2RAB9ACASP3
Methane SCHEMBL28094000 0.67 GRIA1 (0.34) NPC1SMN1; SMN2RAB9ACASP3SENP8
SCHEMBL7833158 0.66 CYP1A2 (0.37) TSHRALDH1A1HSD17B10TP53CYP1A2
SCHEMBL28430350 0.65 ALDH1A1 (0.34) TSHRALDH1A1SMN1; SMN2MAPTHSD17B10
SCHEMBL28963193 0.65 NPC1 (0.32) TSHRNPC1SMN1; SMN2RAB9ACASP3
SCHEMBL7922195 0.65 ADORA2A (0.37) NR1H4NPSR1GAAALDH1A1SMN1; SMN2
SCHEMBL8775987 0.64 MYC (0.33) LMNAALDH1A1AKR1B1MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001766-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2001-04-04 EP disclosed
EP-1001766-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999001127-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-01-14 WO disclosed