SCHEMBL7913508

SCHEMBL7913508

CC1=C(c2ccccc2)C=CC(C(=O)O)(c2noc(C)n2)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.38
ADORA1 P30542 4/20 0.38
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PLK1 P53350 1/20 0.33
MAPT P10636 4/20 0.33
TP53 P04637 3/20 0.33
CHEK1 O14757 1/20 0.33
NTRK1 P04629 1/20 0.33
PIM1 P11309 1/20 0.33
CDK2 P24941 1/20 0.33
CSNK2A1 P68400 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MGLL Q99685 1/20 0.32
POLB P06746 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7922195 0.91 ADORA2A (0.37) ADORA2AADORA1L3MBTL1ALDH1A1NPSR1
SCHEMBL27478872 0.80 ALDH1A1 (0.35) ALDH1A1NPSR1HPGDSMN1; SMN2KDM4E
SCHEMBL27478874 0.80 RAB9A (0.37) ALDH1A1SMN1; SMN2MAPTTP53KDM4E
SCHEMBL27494961 0.77
SCHEMBL27479658 0.75 KDM4E (0.33) ALDH1A1MAPTKDM4E
SCHEMBL27478044 0.75 NPC1 (0.35) ALDH1A1NPSR1MAPTKDM4EGAA
Oxalic Acid SCHEMBL7920408 0.73 HTR1D (0.52) ALDH1A1HPGDMAPTTP53KDM4E
SCHEMBL7922225 0.71 NR1H4 (0.39) L3MBTL1ALDH1A1NPSR1SMN1; SMN2MAPT
SCHEMBL27478043 0.71 HDAC4 (0.35) NTRK1KDM4E
SCHEMBL30161783 0.71 KDM4E (0.33) ALDH1A1HPGDSMN1; SMN2MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001766-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2001-04-04 EP disclosed
EP-1001766-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999001127-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-01-14 WO disclosed