SCHEMBL7922504

SCHEMBL7922504

COC(=O)CC1Nc2ccc(C(=O)N3CCC(C4CCN(C(=O)OCc5ccccc5)CC4)CC3)cc2CNC1=O

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 9/20 0.48
ITGA2B P08514 6/20 0.48
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
FLT3 P36888 1/20 0.42
ITGAV P06756 5/20 0.41
ENPP2 Q13822 1/20 0.41
ATXN2 Q99700 1/20 0.41
GRIN2B Q13224 4/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
GLA P06280 1/20 0.40
CYP2C19 P33261 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7922603 0.92 ITGB3 (0.56) ITGB3ITGA2BSMN1; SMN2NPC1RAB9A
SCHEMBL7922626 0.87 ITGB3 (0.64) ITGB3ITGA2BHTTITGAV
SCHEMBL7916977 0.79 ITGB3 (0.74) ITGB3ITGA2BITGAV
SCHEMBL8144896 0.77 ITGB3 (0.70) ITGB3ITGA2BITGAV
SCHEMBL7910269 0.77 ITGB3 (0.70) ITGB3ITGA2BITGAV
SCHEMBL7078802 0.76 ITGB3 (0.49) ITGB3ITGA2BITGAV
SCHEMBL8525426 0.72 ITGB3 (0.65) ITGB3ITGA2BITGAV
SCHEMBL8194605 0.72 ITGB3 (0.82) ITGB3ITGA2BITGAV
SCHEMBL8525635 0.71 JAK2 (0.46) ITGB3HTTSMN1; SMN2NPC1RAB9A
SCHEMBL7401262 0.70 ITGB3 (0.42) ITGB3HTTITGAVGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6225465-B1 REACTING BENZOAZEPINE OR BENZODIAZEPINE DERIVATIVE WITH PROTECTED AMINE IN PRESENCE OF PALLADIUM CATALYST IN PRESENCE OF CARBON MONOXIDE, REMOVING PROTECTING GROUPS SMITHKLINE BEECHAM PLC (GB) 2001-05-01 US disclosed
EP-1019383-A2 PROCESS FOR THE AMINOCARBONYLATION OF BENZAZEPINES AND BENZODIAZEPINES SMITHKLINE BEECHAM PLC (GB) 2000-07-19 EP disclosed
EP-0964928-A1 ENZYMATIC RESOLUTION OF BENZODIAZEPINE-ACETIC ACID ESTERS WITH A LIPASE SMITHKLINE BEECHAM PLC (GB) 1999-12-22 EP disclosed
WO-1998029561-A1 ENZYMATIC RESOLUTION OF BENZODIAZEPINE-ACETIC ACID ESTERS WITH A LIPASE SMITHKLINE BEECHAM PLC (GB) 1998-07-09 WO disclosed
WO-1997024336-A2 PROCESS FOR THE AMINOCARBONYLATION OF BENZAZEPINES AND BENZODIAZEPINES SMITHKLINE BEECHAM PLC (GB) 1997-07-10 WO disclosed