SCHEMBL8525635

SCHEMBL8525635

COC(=O)CC1Nc2ccccc2CNC1=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.46
HSD17B10 Q99714 7/20 0.45
HTT P42858 2/20 0.45
EGFR P00533 1/20 0.44
KDM4E B2RXH2 10/20 0.43
ALDH1A1 P00352 9/20 0.43
MAPT P10636 6/20 0.43
HPGD P15428 4/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
TP53 P04637 2/20 0.43
TSHR P16473 2/20 0.43
GLA P06280 2/20 0.43
LMNA P02545 1/20 0.43
GAA P10253 2/20 0.41
ITGB3 P05106 2/20 0.41
ITGAV P06756 2/20 0.41
RAB9A P51151 2/20 0.40
MAPK1 P28482 2/20 0.40
ALOX15 P16050 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8468698 0.87 KDM4E (0.44) HSD17B10HTTKDM4EALDH1A1MAPT
SCHEMBL7401262 0.84 ITGB3 (0.42) JAK2HSD17B10HTTEGFRKDM4E
SCHEMBL7916963 0.83 ITGB3 (0.51) HSD17B10HTTEGFRKDM4EALDH1A1
SCHEMBL7916970 0.83 ITGB3 (0.51) HSD17B10HTTEGFRKDM4EALDH1A1
SCHEMBL7917615 0.83 ITGB3 (0.41) JAK2HSD17B10HTTEGFRKDM4E
SCHEMBL8399397 0.82 EPHX2 (0.44) HSD17B10HTTKDM4EALDH1A1MAPT
SCHEMBL7078802 0.82 ITGB3 (0.49) JAK2KDM4EMAPTITGB3ITGAV
SCHEMBL4428402 0.79 KDM4E (0.63) HSD17B10HTTKDM4EALDH1A1MAPT
SCHEMBL644092 0.79 KDM4E (0.63) HSD17B10HTTKDM4EALDH1A1MAPT
SCHEMBL7399767 0.79 ALDH1A1 (0.40) ALDH1A1MAPTLMNAGAAITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0964928-A1 ENZYMATIC RESOLUTION OF BENZODIAZEPINE-ACETIC ACID ESTERS WITH A LIPASE SMITHKLINE BEECHAM PLC (GB) 1999-12-22 EP disclosed
WO-1998029561-A1 ENZYMATIC RESOLUTION OF BENZODIAZEPINE-ACETIC ACID ESTERS WITH A LIPASE SMITHKLINE BEECHAM PLC (GB) 1998-07-09 WO disclosed