SCHEMBL7923133

SCHEMBL7923133

COc1ccc(C(=O)C(C)=NO)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.67
CES1 P23141 2/20 0.67
MAPT P10636 4/20 0.62
SMN1; SMN2 Q16637 3/20 0.62
POLB P06746 1/20 0.62
ALDH1A1 P00352 2/20 0.57
CA1 P00915 6/20 0.53
CA2 P00918 6/20 0.53
PARP1 P09874 1/20 0.52
PARP10 Q53GL7 1/20 0.52
PARP2 Q9UGN5 1/20 0.52
PARP4 Q9UKK3 1/20 0.52
PLK1 P53350 1/20 0.48
MEN1 O00255 2/20 0.48
LMNA P02545 2/20 0.48
KMT2A Q03164 2/20 0.48
NPSR1 Q6W5P4 2/20 0.48
GAA P10253 1/20 0.48
GFER P55789 1/20 0.48
KDM4E B2RXH2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11370460 1.00 CES2 (0.67) CES2CES1MAPTSMN1; SMN2POLB
SCHEMBL10810096 1.00 CES2 (0.67) CES2CES1MAPTSMN1; SMN2POLB
SCHEMBL4711175 0.81 CES2 (0.62) CES2CES1MAPTSMN1; SMN2POLB
SCHEMBL4711178 0.81 CES2 (0.62) CES2CES1MAPTSMN1; SMN2POLB
SCHEMBL557152 0.81 CES2 (1.00) CES2CES1MAPTCA1CA2
SCHEMBL14507040 0.81 CES2 (1.00) CES2CES1MAPTCA1CA2
SCHEMBL11489865 0.80 PARP10 (0.56) MAPTSMN1; SMN2POLBALDH1A1PARP10
SCHEMBL11714663 0.80 PARP10 (0.53) CES2CES1MAPTSMN1; SMN2POLB
SCHEMBL11714645 0.80 PARP10 (0.53) CES2CES1MAPTSMN1; SMN2POLB
SCHEMBL11489871 0.80 PARP10 (0.56) MAPTSMN1; SMN2POLBALDH1A1PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6225463-B1 REACTING S-AMINE COMPOUND WITH AN ALDEHYDE; REACTING WITH ACYL CHLORIDE IN PRESENCE OF TRIETHYLAMINE TO FORM DIASTEREOISOMERIC BETA-LACTAMS; SEPARATION; TREATING WITH CERIUM AMMONIUM NITRATE AND ACETONITRILE AND WATER PHARMACHEMIE B.V. (NL) 2001-05-01 US disclosed
EP-0933360-A1 Synthesis of new beta-lactams PHARMACHEMIE B.V. (NL) 1999-08-04 EP disclosed
EP-0077983-B1 TRIAZINE DERIVATIVES, PROCESSES FOR PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-04-29 EP disclosed
EP-0077983-A1 Triazine derivatives, processes for preparation thereof and pharmaceutical compositions comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-05-04 EP disclosed
US-4293552-A Novel 1-(mono-o-substituted benzoyl)-3-(substituted pyrazinyl) ureas ELI LILLY AND COMPANY (US) 1981-10-06 US disclosed
US-4229579-A OPTICAL BRIGHTENERS BAYER AKTIENGESELLSCHAFT (DE) 1980-10-21 US disclosed
US-4160834-A INSECTICIDES ELI LILLY AND COMPANY (US) 1979-07-10 US disclosed
US-4144243-A OPTICAL BRIGHTENERS FOR TEXTILES AND LACQUEARS BAYER AKTIENGESELLSCHAFT (DE) 1979-03-13 US disclosed
US-4083977-A Novel insecticidal 1-(substituted benzoyl)-3-(substituted pyrazinyl)ureas ELI LILLY AND COMPANY (US) 1978-04-11 US disclosed