SCHEMBL7927451

SCHEMBL7927451

CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)NC(c1cccc(Cl)c1)c1cccc(OCc2ccccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.49
KLK7 P49862 1/20 0.47
CTSL P07711 1/20 0.46
BACE1 P56817 7/20 0.44
CTSS P25774 2/20 0.43
CTSK P43235 2/20 0.43
PSMB1 P20618 1/20 0.43
PSMB8 P28062 1/20 0.43
PSMB9 P28065 1/20 0.43
PSMB5 P28074 1/20 0.43
REN P00797 1/20 0.43
S1PR3 Q99500 1/20 0.43
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
CA2 P00918 1/20 0.42
PKM P14618 1/20 0.42
BACE2 Q9Y5Z0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7719347 1.00 KLK5 (0.49) KLK5KLK7CTSLBACE1CTSS
Methane SCHEMBL7719349 0.89 CTSL (0.47) CTSLCTSSCTSKPSMB1PSMB8
SCHEMBL7718473 0.82 KLK5 (0.54) KLK5KLK7BACE1CTSSCTSK
SCHEMBL5570005 0.77 KLK5 (0.56) KLK5KLK7BACE1CTSSCTSK
SCHEMBL5570008 0.77 KLK5 (0.56) KLK5KLK7BACE1CTSSCTSK
SCHEMBL7936792 0.76 KLK5 (0.50) KLK5KLK7BACE1CTSSCTSK
SCHEMBL27983817 0.75 KMT2A (0.51)
SCHEMBL6555039 0.75 HDAC4 (0.55) KLK5CTSLCTSSCTSKKDM4E
SCHEMBL15783809 0.74 CHRM3 (0.49) CTSSCTSKPSMB1PSMB8PSMB9
SCHEMBL14166143 0.74 CHRM3 (0.61) PSMB1PSMB8PSMB9PSMB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001017992-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed