SCHEMBL7936792

SCHEMBL7936792

CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccc2ccc(OCc3ccccc3)cc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.50
KLK7 P49862 1/20 0.48
HDAC1 Q13547 5/20 0.47
HDAC2 Q92769 2/20 0.47
PTPN1 P18031 1/20 0.47
KDM4E B2RXH2 3/20 0.46
ALDH1A1 P00352 3/20 0.46
MAPT P10636 1/20 0.46
HDAC4 P56524 4/20 0.45
HDAC6 Q9UBN7 4/20 0.45
CTSS P25774 3/20 0.45
CTSK P43235 3/20 0.45
LMNA P02545 2/20 0.45
CTSB P07858 1/20 0.45
THRB P10828 1/20 0.45
HPGD P15428 1/20 0.45
HDAC3 O15379 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7718633 0.84 ALDH1A1 (0.47) KLK5HDAC1HDAC2KDM4EALDH1A1
SCHEMBL5570008 0.83 KLK5 (0.56) KLK5KLK7CTSSCTSKHDAC8
SCHEMBL5570005 0.83 KLK5 (0.56) KLK5KLK7CTSSCTSKHDAC8
SCHEMBL4485886 0.83 PLAU (0.52) HDAC1PTPN1
SCHEMBL7718473 0.81 KLK5 (0.54) KLK5KLK7CTSSCTSKBACE1
SCHEMBL6432668 0.78 HDAC1 (0.46) HDAC1PTPN1MEN1KMT2A
SCHEMBL11036298 0.77 HDAC4 (0.53) KLK5KLK7HDAC1HDAC2KDM4E
SCHEMBL5570659 0.77 ALDH1A1 (0.49) KLK5KLK7HDAC1KDM4EALDH1A1
SCHEMBL5570666 0.77 ALDH1A1 (0.49) KLK5KLK7HDAC1KDM4EALDH1A1
SCHEMBL7927451 0.76 KLK5 (0.49) KLK5KLK7KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001017992-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed