SCHEMBL7928394

SCHEMBL7928394

COC(=O)c1ccc(C#Cc2ccc(OCc3ccccc3)cc2)cc1O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.59
PTPN11 Q06124 2/20 0.54
PTPN1 P18031 1/20 0.54
PTPN6 P29350 1/20 0.54
APP P05067 1/20 0.53
LMNA P02545 2/20 0.52
HPGD P15428 1/20 0.52
ACACB O00763 1/20 0.50
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
MCL1 Q07820 1/20 0.49
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48
PDK2 Q15119 1/20 0.48
PDK4 Q16654 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL629952 0.88 MAOB (0.74) MAOBAPPLMNAHPGDNPC1
SCHEMBL15942083 0.86 PTPN11 (0.56) PTPN11LMNASMN1; SMN2CA12CA1
SCHEMBL1391085 0.85 PTPN1 (0.51) MAOBPTPN11PTPN1PTPN6APP
Methyl 2,4-Dihydroxybenzoate SCHEMBL5199862 0.85 MAOB (0.68) MAOBAPPLMNAHPGDNPC1
SCHEMBL23405322 0.85 FFAR4 (0.53) MAOBPTPN11PTPN1PTPN6LMNA
SCHEMBL29820043 0.81 CA12 (0.65) PTPN11LMNAHPGDNPC1SMN1; SMN2
SCHEMBL15603819 0.81 CA12 (0.65) PTPN11LMNAHPGDNPC1SMN1; SMN2
SCHEMBL15603818 0.80 FFAR4 (0.48) MAOBPTPN11PTPN1PTPN6LMNA
SCHEMBL3712925 0.80 ACACB (0.58) MAOBPTPN11PTPN1PTPN6LMNA
SCHEMBL710202 0.79 MAOB (0.63) MAOBAPPLMNAHPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2351743-A1 BICYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-08-03 EP disclosed
WO-2010050445-A1 BICYCLIC COMPOUND 武田薬品工業株式会社 (JP) 2010-05-06 WO disclosed