SCHEMBL7928459

SCHEMBL7928459

CCCOCCOc1ccc2cc(OB(O)O)oc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 6/20 0.48
CA12 O43570 5/20 0.48
CA1 P00915 5/20 0.48
CA6 P23280 3/20 0.48
CA7 P43166 3/20 0.48
CA14 Q9ULX7 3/20 0.48
CA5B Q9Y2D0 3/20 0.48
CA2 P00918 2/20 0.48
CA5A P35218 2/20 0.48
CA4 P22748 2/20 0.45
CA3 P07451 1/20 0.45
KDM4E B2RXH2 2/20 0.41
MAPK1 P28482 2/20 0.41
NPC1 O15118 2/20 0.41
MAPT P10636 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GLA P06280 2/20 0.41
MAOA P21397 2/20 0.41
MAOB P27338 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7929600 0.92 CA9 (0.56) CA9CA12CA1CA6CA7
SCHEMBL7929537 0.90 MAOB (0.41) CA9CA12CA1CA6CA7
SCHEMBL7931672 0.82 MAOB (0.46) CA9CA12CA1CA6CA7
SCHEMBL7929599 0.81 CA9 (0.58) CA9CA12CA1CA6CA7
SCHEMBL7931713 0.78 CA9 (0.38) CA9CA12CA1CA6CA7
SCHEMBL5657236 0.75 LMNA (0.45) KDM4EMAPK1MAPTSMN1; SMN2ALDH1A1
SCHEMBL7929502 0.74 CNR2 (0.41) CA9CA12CA1CA2KDM4E
SCHEMBL28632856 0.73 CA9 (0.58) CA9CA12CA1CA6CA7
SCHEMBL7221364 0.73 ALDH1A1 (0.48) KDM4EMAPK1MAPTALDH1A1L3MBTL1
SCHEMBL7934233 0.72 KDM4E (0.40) KDM4EMAPK1MAPTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed