SCHEMBL7928499

SCHEMBL7928499

CCCOC(C)Oc1cccc2ccoc12

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.32
EGLN1 Q9GZT9 1/20 0.32
HTR1A P08908 1/20 0.31
SLC6A4 P31645 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3789173 0.79 MCHR1 (0.49) MCHR1MEN1ALDH1A1LMNAHPGD
SCHEMBL3789397 0.79 MCHR1 (0.46) MCHR1HTR1ASLC6A4
SCHEMBL3799434 0.78 MCHR1 (0.44) MCHR1MEN1ALDH1A1LMNAHPGD
SCHEMBL3795511 0.74 MCHR1 (0.48) MCHR1HTR1ASLC6A4CNR2
SCHEMBL7929500 0.74 CNR2 (0.36) ALDH1A1LMNAKMT2ACNR2
SCHEMBL7928500 0.74 NCF1 (0.40) MCHR1HTR1ASLC6A4MEN1ALDH1A1
SCHEMBL11849207 0.72 KMT2A (0.40) MEN1ALDH1A1LMNAHPGDKMT2A
SCHEMBL7929506 0.72 CNR2 (0.38) MEN1ALDH1A1LMNAKMT2ACNR2
SCHEMBL11810492 0.72 MEN1 (0.33) SLC6A4MEN1ALDH1A1LMNAHPGD
SCHEMBL3796715 0.72 ADORA3 (0.49) MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed