SCHEMBL7928689

SCHEMBL7928689

Cc1ccnc(NN=C(c2ccccc2)c2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
LMNA P02545 1/20 0.53
HTT P42858 1/20 0.53
RAB9A P51151 3/20 0.52
NPC1 O15118 2/20 0.52
NOS2 P35228 1/20 0.49
ATM Q13315 1/20 0.48
KDR P35968 2/20 0.46
MAP4K4 O95819 1/20 0.46
ABL1 P00519 1/20 0.46
LCK P06239 1/20 0.46
FYN P06241 1/20 0.46
IGF1R P08069 1/20 0.46
LTK P29376 1/20 0.46
MAP2K2 P36507 1/20 0.46
MAPK8 P45983 1/20 0.46
MAPK9 P45984 1/20 0.46
CLK2 P49760 1/20 0.46
GSK3A P49840 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20101033 0.89 KDM4E (0.58) ALDH1A1SMN1; SMN2LMNAHTTRAB9A
SCHEMBL10289446 0.81 KDM4E (0.52) ALDH1A1SMN1; SMN2LMNAHTTRAB9A
SCHEMBL2564755 0.81 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2LMNAHTTRAB9A
SCHEMBL2564746 0.81 NOS3 (0.51) ALDH1A1SMN1; SMN2LMNAHTTRAB9A
SCHEMBL25203872 0.79 SMN1; SMN2 (0.46) ALDH1A1SMN1; SMN2LMNAHTTRAB9A
SCHEMBL15267189 0.78 KDM4E (0.58) ALDH1A1SMN1; SMN2LMNAHTTRAB9A
SCHEMBL1195267 0.75 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2LMNAHTTRAB9A
SCHEMBL25241674 0.75 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2LMNAHTTRAB9A
SCHEMBL25224389 0.75 MAPT (0.51) ALDH1A1SMN1; SMN2LMNAHTTRAB9A
SCHEMBL15279086 0.74 KDM4E (0.48) ALDH1A1SMN1; SMN2LMNAHTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102026985-A Quinazoline derivatives as RAF kinase modulators and methods and uses thereof AMBIT BIOSCIENCES CORPORATON 2011-04-20 CN disclosed
WO-2010076525-A1 DERIVATIVES OF 2-PYRIDIN-2-YL-PYRAZOL-3(2H)-ONE, PREPARATION AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2010-07-08 WO disclosed
WO-2010076524-A2 DERIVATIVES OF 2-PYRIDIN-2-YL-PYRAZOL-3(2H)-ONE, PREPARATION AND THERAPEUTIC USE THEREOF AS HIF ACTIVATORS SANOFI-AVENTIS (FR) 2010-07-08 WO disclosed