SCHEMBL7929311

SCHEMBL7929311

Cc1ccc(NC(=O)c2cn3cc(C)nc3c(-c3cccc(Cl)c3)n2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 2/20 0.47
CNR2 P34972 2/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
HPGD P15428 1/20 0.43
EGLN1 Q9GZT9 2/20 0.43
TP53 P04637 2/20 0.43
GAA P10253 1/20 0.43
GHSR Q92847 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KDM5B Q9UGL1 1/20 0.42
CNR1 P21554 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7932093 0.86 ROCK1 (0.43) ROCK1CNR2MEN1KMT2APOLB
SCHEMBL7934185 0.86 MAPT (0.54) MEN1KMT2APOLBMAPTSMN1; SMN2
SCHEMBL7930900 0.85 MAPT (0.49) ROCK1CNR2MEN1KMT2APOLB
SCHEMBL7928073 0.81 TRPV1 (0.42)
SCHEMBL7931544 0.75 CNR2 (0.50) CNR2MEN1KMT2APOLBMAPT
SCHEMBL7930354 0.73 SMN1; SMN2 (0.47) CNR2MEN1KMT2APOLBMAPT
SCHEMBL1937367 0.73 KDR (0.56) CNR2MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL23928620 0.72 MEN1 (0.81) MEN1KMT2APOLBMAPTSMN1; SMN2
SCHEMBL3367808 0.70 EGLN1 (0.72) CNR2MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL13500816 0.70 SLC2A1 (0.71) CNR2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed