SCHEMBL7932093

SCHEMBL7932093

Cc1cn2cc(C(=O)Nc3ccc(N)nc3)nc(-c3cccc(Cl)c3)c2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.43
JAK2 O60674 5/20 0.43
CYP3A4 P08684 1/20 0.43
ATR Q13535 1/20 0.41
BACE1 P56817 1/20 0.40
KCNQ3 O43525 1/20 0.40
KCNQ2 O43526 1/20 0.40
KCNE1 P15382 1/20 0.40
KCNQ1 P51787 1/20 0.40
CNR2 P34972 2/20 0.39
CDK8 P49336 2/20 0.39
MAPK10 P53779 1/20 0.39
POLB P06746 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
JAK1 P23458 2/20 0.38
CYP1A2 P05177 1/20 0.38
TYK2 P29597 1/20 0.38
JAK3 P52333 1/20 0.38
EGLN1 Q9GZT9 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7929311 0.86 ROCK1 (0.47) ROCK1CYP3A4CNR2POLBMEN1
SCHEMBL7934185 0.85 MAPT (0.54) POLBMEN1KMT2ATP53MAPT
SCHEMBL7929299 0.84 KCNQ3 (0.43) JAK2CYP3A4ATRKCNQ3KCNQ2
SCHEMBL7928073 0.84 TRPV1 (0.42)
SCHEMBL7930900 0.79 MAPT (0.49) ROCK1CNR2POLBMEN1KMT2A
SCHEMBL7932092 0.73 KCNQ3 (0.45) JAK2CYP3A4ATRKCNQ3KCNQ2
SCHEMBL7930350 0.69 POLB (0.51) POLBMEN1KMT2ATP53MAPT
SCHEMBL7921912 0.69
SCHEMBL7931544 0.69 CNR2 (0.50) ATRCNR2POLBMEN1KMT2A
SCHEMBL3378478 0.68 DHFR (0.39) BACE1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed