SCHEMBL7930064

SCHEMBL7930064

Clc1ccc(C(Cl)(Cl)Cl)c(C(Cl)(Cl)Cl)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.44
CYP3A4 P08684 2/20 0.44
MAPK1 P28482 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
NOTUM Q6P988 1/20 0.31
LMNA P02545 1/20 0.30
PNMT P11086 1/20 0.30
CYP2A6 P11509 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10999631 0.82 TSHR (0.46) TSHRCYP3A4MAPK1TDP1NOTUM
SCHEMBL28645554 0.81 TSHR (0.40) TSHRCYP3A4MAPK1TDP1NOTUM
SCHEMBL6415524 0.79 TSHR (0.48) TSHRCYP3A4MAPK1TDP1LMNA
SCHEMBL11601275 0.75 TSHR (0.44) TSHRCYP3A4MAPK1TDP1
SCHEMBL10493705 0.73 TSHR (0.34) TSHRCYP3A4MAPK1NOTUMLMNA
SCHEMBL10493736 0.73 TSHR (0.43) TSHRCYP3A4MAPK1TDP1NOTUM
SCHEMBL8664297 0.73 TSHR (0.43) TSHRCYP3A4MAPK1TDP1NOTUM
SCHEMBL11003720 0.72 TSHR (0.50) TSHRCYP3A4MAPK1TDP1LMNA
SCHEMBL2262591 0.69 TSHR (0.46) TSHRCYP3A4MAPK1TDP1LMNA
SCHEMBL8846801 0.68 TSHR (0.43) TSHRCYP3A4MAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6201152-B1 HEATING MIXTURE OF METHYL-3,5-DICHLORO-4-METHYLBENZOATE AND ALPHA,ALPHA,ALPHA-TRICHLOROMETHYLBENZENE IN PRESENCE OF AMMONIUM MOLYBDATE CATALYST OCCIDENTAL CHEMICAL CORPORATION 2001-03-13 US claimed
US-4080378-A REACTING A CARBOXYLIC ACID ESTER WITH A TRICHLOROMETHYL SUBSTITUTED AROMATIC COMPOUND IN THE PRESENCE OF A MOLYBDENUM CATALYST DYNAMIT NOBEL AKTIENGESELLSCHAFT (DT) 1978-03-21 US claimed
US-6201152-B1 HEATING MIXTURE OF METHYL-3,5-DICHLORO-4-METHYLBENZOATE AND ALPHA,ALPHA,ALPHA-TRICHLOROMETHYLBENZENE IN PRESENCE OF AMMONIUM MOLYBDATE CATALYST OCCIDENTAL CHEMICAL CORPORATION 2001-03-13 US disclosed
US-4104300-A MOLYBDENUM CATALYST, COMPLEXING AGENT DYNAMIT NOBEL AKTIENGESELLSCHAFT (DE) 1978-08-01 US disclosed
US-4080378-A REACTING A CARBOXYLIC ACID ESTER WITH A TRICHLOROMETHYL SUBSTITUTED AROMATIC COMPOUND IN THE PRESENCE OF A MOLYBDENUM CATALYST DYNAMIT NOBEL AKTIENGESELLSCHAFT (DT) 1978-03-21 US disclosed