SCHEMBL7930732

SCHEMBL7930732

Cc1cn2cc(C(=O)Nc3ccccn3)cc(-c3cccc(Cl)c3)c2n1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.53
GRM5 P41594 3/20 0.49
ALDH1A1 P00352 3/20 0.48
SIRT2 Q8IXJ6 1/20 0.45
KCNMA1 Q12791 1/20 0.45
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
TDP1 Q9NUW8 1/20 0.43
MAPK14 Q16539 1/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
TP53 P04637 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KDM4E B2RXH2 1/20 0.42
JAK2 O60674 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7931544 0.86 CNR2 (0.50) CNR2GRM5ALDH1A1NPC1RAB9A
SCHEMBL7930354 0.84 SMN1; SMN2 (0.47) CNR2GRM5ALDH1A1SIRT2KCNMA1
SCHEMBL7934025 0.84 NPC1 (0.49) GRM5ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL7930350 0.82 POLB (0.51) SIRT2KCNMA1NPC1RAB9AMEN1
SCHEMBL7922479 0.81 JAK2 (0.46) GRM5MEN1KMT2AL3MBTL1JAK2
SCHEMBL7929316 0.81 GCK (0.62) GRM5ALDH1A1NPC1RAB9AMEN1
SCHEMBL7929299 0.80 KCNQ3 (0.43) GRM5MAPK14JAK2
SCHEMBL3377871 0.79 MAPK14 (0.46) GRM5ALDH1A1NPC1RAB9AKMT2A
SCHEMBL7921912 0.79
SCHEMBL7930895 0.77 PSMD14 (0.43) CNR2GRM5ALDH1A1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed