SCHEMBL7930987

SCHEMBL7930987

CC(C)C[C@@H](C(=O)NN(CC(C)C)C(=O)CNC(N)=O)[C@H](CC=Cc1ccccc1)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 1/20 0.55
GRIK1 P39086 4/20 0.37
GRIK2 Q13002 4/20 0.37
HTR2A P28223 3/20 0.35
CTSC P53634 1/20 0.34
FCER2 P06734 1/20 0.33
MASP2 O00187 1/20 0.33
MMP2 P08253 1/20 0.32
MMP3 P08254 1/20 0.32
MMP7 P09237 1/20 0.32
LTA4H P09960 1/20 0.32
ANPEP P15144 1/20 0.32
EPOR P19235 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981779 0.94 ADAM17 (0.64) ADAM17FCER2MMP2MMP3MMP7
SCHEMBL6939982 0.87 ADAM17 (0.59) ADAM17GRIK1GRIK2HTR2ACTSC
SCHEMBL6983321 0.85 ADAM17 (0.65) ADAM17FCER2MMP2MMP3MMP7
SCHEMBL6945913 0.84 ADAM17 (0.63) ADAM17GRIK1GRIK2HTR2ACTSC
SCHEMBL6984710 0.82 ADAM17 (0.45) ADAM17
Hydrochloric Acid SCHEMBL6982517 0.82 ADAM17 (0.66) ADAM17FCER2MMP2MMP3MMP7
SCHEMBL7931029 0.82 ADAM17 (0.57) ADAM17GRIK1GRIK2HTR2ACTSC
SCHEMBL6986418 0.81 ADAM17 (0.70) ADAM17FCER2MMP2MMP3MMP7
SCHEMBL6937771 0.81 ADAM17 (0.69) ADAM17FCER2MMP2MMP3MMP7
SCHEMBL6942575 0.79 ADAM17 (0.73) ADAM17FCER2MMP2MMP3MMP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6239151-B1 TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISEASES, OSTEOARTHRITIS, RESPIRATORY DISEASES, TUMORS, CACHEXIA, CARDIOVASCULAR DISEASES, FEVER, HAEMORRHAGE AND SEPSIS, HYDRAZINE DERIVATIVES, HOFFMANN-LA ROCHE INC. 2001-05-29 US disclosed