SCHEMBL7932450

SCHEMBL7932450

N#Cc1ccccc1C1CCC(NCCN)CC1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 6/20 0.48
KDM4E B2RXH2 1/20 0.45
SMYD3 Q9H7B4 1/20 0.40
HCRTR2 O43614 2/20 0.39
DRD4 P21917 1/20 0.38
ADRA1A P35348 2/20 0.36
SLC6A4 P31645 1/20 0.35
EZH2 Q15910 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7934160 0.99 OPRL1 (0.47) OPRL1KDM4ESMYD3HCRTR2DRD4
Hydrochloric Acid SCHEMBL7936704 0.99 OPRL1 (0.47) OPRL1KDM4ESMYD3HCRTR2DRD4
Hydrochloric Acid SCHEMBL7934158 0.99 OPRL1 (0.47) OPRL1KDM4ESMYD3HCRTR2DRD4
SCHEMBL7994302 0.82 OPRL1 (0.44) OPRL1KDM4EHCRTR2DRD4ADRA1A
SCHEMBL8003101 0.81 DRD4 (0.42) OPRL1KDM4EHCRTR2DRD4ADRA1A
SCHEMBL7106832 0.80 GRIN2B (0.49) OPRL1KDM4ESLC6A4
SCHEMBL3167985 0.79 ADRA1A (0.49) OPRL1KDM4EHCRTR2DRD4ADRA1A
SCHEMBL29580963 0.79 ADRA1A (0.49) OPRL1KDM4EHCRTR2DRD4ADRA1A
SCHEMBL8178976 0.77 OPRL1 (0.43) OPRL1KDM4EHCRTR2DRD4ADRA1A
SCHEMBL7714987 0.76 KDM4E (0.44) KDM4EDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235759-B1 BENIGN PROSTATIC HYPERPLASIA; HYPOTENSIVE AGENTS MERCK & CO., INC. 2001-05-22 US disclosed
WO-2000025782-A1 DIHYDROPYRIDINONES AND PYRROLINONES USEFUL AS ALPHA 1A ADRENOCEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2000-05-11 WO disclosed