SCHEMBL7932694

SCHEMBL7932694

FC(F)(F)c1ccc(-c2ccccc2/C=C/I)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.47
NR1H3 Q13133 1/20 0.41
BACE1 P56817 2/20 0.40
ALDH1A1 P00352 2/20 0.39
TSHR P16473 1/20 0.39
CYP1A2 P05177 2/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
CYP2C19 P33261 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MAOB P27338 2/20 0.37
CYP1A1 P04798 1/20 0.37
CYP1B1 Q16678 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
GAA P10253 1/20 0.36
CHUK O15111 1/20 0.36
TXNRD1 Q16881 1/20 0.36
NOX4 Q9NPH5 1/20 0.36
JAK2 O60674 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7932699 1.00 KIF11 (0.47) KIF11NR1H3BACE1ALDH1A1TSHR
SCHEMBL28717114 0.81 NR1H3 (0.54) KIF11NR1H3BACE1ALDH1A1TSHR
SCHEMBL29507315 0.81 NR1H3 (0.54) KIF11NR1H3BACE1ALDH1A1TSHR
SCHEMBL7930951 0.80 SLC6A4 (0.41) BACE1
SCHEMBL7930955 0.80 SLC6A4 (0.41) BACE1
SCHEMBL7935558 0.79 BACE1 (0.46) BACE1ALDH1A1HSD17B10
SCHEMBL7935560 0.79 BACE1 (0.46) BACE1ALDH1A1HSD17B10
SCHEMBL8175555 0.79 BACE1 (0.46) BACE1ALDH1A1HSD17B10
SCHEMBL416843 0.79 KIF11 (0.50) KIF11NR1H3BACE1ALDH1A1TSHR
Ammonia Solution, Strong SCHEMBL6558306 0.77 KIF11 (0.48) KIF11NR1H3BACE1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0879814-B1 Triaromatic compounds, compositions containing them and uses thereof CT INTERNAT DE BR RECH S DERMA (FR) 2001-11-28 EP disclosed
US-6150413-A TREATMENT OF DERMATOLOGICAL, RHEUMATIC, RESPIRATORY, CARDIOVASCULAR, BONE AND OPHTHALMOLOGICAL DISORDERS, AS WELL AS MAMMALIAN SKIN AND HAIR CONDITIONS; 4-(4-(BIPHENYL-2-YL)BUT-3-EN-1-YNYL)BENZOIC ACID, FOR EXAMPLE CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (FR) 2000-11-21 US disclosed
EP-0879814-A1 Triaromatic compounds, compositions containing them and uses thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (C.I.R.D. GALDERMA) (FR) 1998-11-25 EP disclosed