SCHEMBL7932790

SCHEMBL7932790

Cc1cc(Cl)ccc1OC(=O)C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.57
HTR2A P28223 1/20 0.57
HTR2C P28335 1/20 0.57
HTR2B P41595 1/20 0.57
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
HIF1A Q16665 1/20 0.50
MRGPRX4 Q96LA9 2/20 0.47
NPSR1 Q6W5P4 2/20 0.47
KDM4E B2RXH2 3/20 0.47
TP53 P04637 1/20 0.47
ALOX15 P16050 1/20 0.47
ALDH1A1 P00352 2/20 0.46
HTT P42858 3/20 0.45
MAPT P10636 3/20 0.45
LMNA P02545 5/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
HPGD P15428 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29131709 0.86 TSHR (0.54) TSHRHTR2AHTR2CHTR2BCYP1A2
SCHEMBL6273604 0.85 TSHR (0.60) TSHRHTR2AHTR2CHTR2BCYP1A2
Hydrochloric Acid SCHEMBL11854026 0.84 TSHR (0.58) TSHRHTR2AHTR2CHTR2BCYP1A2
SCHEMBL27831889 0.81 TDP1 (0.56) TSHRMRGPRX4ALDH1A1MAPTLMNA
SCHEMBL7934361 0.81 L3MBTL1 (0.49) TSHRCYP1A2CYP2C9MRGPRX4NPSR1
SCHEMBL11716516 0.81 TSHR (0.56) TSHRHTR2AHTR2CHTR2BCYP1A2
SCHEMBL132336 0.81 TSHR (0.56) TSHRHTR2AHTR2CHTR2BCYP1A2
SCHEMBL5712913 0.80 TSHR (0.54) TSHRHTR2AHTR2CHTR2BCYP1A2
SCHEMBL13342826 0.79 TSHR (0.57) TSHRHTR2AHTR2CHTR2BCYP1A2
SCHEMBL8766097 0.79 KMT2A (0.56) TSHRHTR2AHTR2CHTR2BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0814074-B1 PROCESS FOR PREPARING DIARYL ESTERS OF OXALIC ACID UBE INDUSTRIES (JP) 2001-03-28 EP disclosed
US-6018072-A SUBJECTING AN ALKYLARYL OXALATE TO A DISPROPORTIONATION REACTION IN THE PRESENCE OF A DISPROPORTIONATION CATALYST TO PRODUCE A DIARYL OXALATE WHILE REMOVING A DIALKYL OXALATE BY-PRODUCT UBE INDUSTRIES, LTD. (JP) 2000-01-25 US disclosed
EP-0814074-A1 PROCESS FOR PREPARING DIARYL ESTERS OF OXALIC ACID UBE INDUSTRIES, LTD. (JP) 1997-12-29 EP disclosed