SCHEMBL7934201

SCHEMBL7934201

OB(O)Oc1ccc(CN2CCOCC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.64
HRH3 Q9Y5N1 5/20 0.59
TSHR P16473 1/20 0.49
HIF1A Q16665 1/20 0.49
EPAS1 Q99814 1/20 0.49
NOS3 P29474 1/20 0.49
NOS1 P29475 1/20 0.49
NOS2 P35228 1/20 0.49
HTT P42858 1/20 0.48
HPGD P15428 1/20 0.48
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48
KCNJ1 P48048 1/20 0.48
KDM4E B2RXH2 1/20 0.47
CACNA1B Q00975 1/20 0.47
APBA1 Q02410 1/20 0.47
SAE1 Q9UBE0 1/20 0.47
UBA2 Q9UBT2 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27993741 0.92 SMN1; SMN2 (0.58) SMN1; SMN2HRH3TSHRHIF1AEPAS1
SCHEMBL28295890 0.85 HRH3 (0.59) HRH3TSHRALDH1A1KDM4E
SCHEMBL28215483 0.84 SIGMAR1 (0.51) SMN1; SMN2HRH3TSHRHTTALDH1A1
SCHEMBL28234040 0.82 KDM4E (0.66) SMN1; SMN2HRH3NOS1HTTHPGD
SCHEMBL28032662 0.81 ALDH1A1 (0.63) HRH3TSHRHPGDALDH1A1LMNA
SCHEMBL15467001 0.80 HRH3 (0.87) SMN1; SMN2HRH3HIF1AEPAS1NOS3
SCHEMBL7931600 0.78 NPC1 (0.61) SMN1; SMN2HRH3TSHRALDH1A1LMNA
SCHEMBL29127455 0.78 HRH3 (0.54) SMN1; SMN2HRH3TSHRALDH1A1LMNA
SCHEMBL2545899 0.78 HRH3 (0.65) SMN1; SMN2HRH3HIF1AEPAS1NOS3
SCHEMBL5755331 0.78 SMN1; SMN2 (1.00) SMN1; SMN2HRH3TSHRHIF1AEPAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104302624-B Antimalarial agent MERCK PATENT GMBH (DE) 2016-01-13 CN disclosed
CN-104302624-A Anti-malarial agents UNIV DUNDEE 2015-01-21 CN disclosed
CN-104080769-A Aryl or heteroaryl substituted benzene compounds EPIZYME INC 2014-10-01 CN disclosed
CN-101094848-B Organic compounds NOVARTIS AG 2013-03-13 CN disclosed
EP-1140896-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 Takeda Chemical Industries, Ltd. (JP) 2001-10-10 EP disclosed
US-6235771-B1 AIDS THERPAY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
WO-2000037455-A1 BENZOTHIEPIN-ANILIDE DERIVATIVES, THEIR PRODUCTION AND THEIR USE FOR ANTAGONIZING CCR-5 TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-06-29 WO disclosed