SCHEMBL7934328

SCHEMBL7934328

COC(=O)Nc1ccc(Nc2ccc(O)cc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.63
GAA P10253 4/20 0.63
LMNA P02545 3/20 0.63
GFER P55789 2/20 0.63
POLB P06746 2/20 0.63
MAPT P10636 6/20 0.55
ALDH1A1 P00352 3/20 0.55
CA12 O43570 2/20 0.55
CA1 P00915 2/20 0.55
CA2 P00918 2/20 0.55
CA7 P43166 2/20 0.55
CA9 Q16790 2/20 0.55
CA14 Q9ULX7 2/20 0.55
MEN1 O00255 1/20 0.55
BRD4 O60885 1/20 0.55
NR1I2 O75469 1/20 0.55
MB P02144 1/20 0.55
CYP1A1 P04798 1/20 0.55
CA3 P07451 1/20 0.55
CYP3A4 P08684 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9089994 0.94 SMN1; SMN2 (0.69) SMN1; SMN2GAALMNAGFERPOLB
SCHEMBL9125125 0.88 SMN1; SMN2 (0.63) SMN1; SMN2GAALMNAGFERPOLB
SCHEMBL9609808 0.85 SMN1; SMN2 (0.82) SMN1; SMN2GAALMNAGFERPOLB
SCHEMBL9479507 0.84 HPGD (0.68) SMN1; SMN2GAALMNAGFERPOLB
SCHEMBL9123962 0.82 SMN1; SMN2 (0.56) SMN1; SMN2GAALMNAGFERPOLB
SCHEMBL22930929 0.79 KMT2A (0.87) SMN1; SMN2LMNAPOLBMAPTALDH1A1
SCHEMBL7251623 0.79 SMN1; SMN2 (0.72) SMN1; SMN2GAALMNAGFERPOLB
SCHEMBL13186585 0.78 LMNA (1.00) SMN1; SMN2GAALMNAGFERPOLB
SCHEMBL17518815 0.77 SMN1; SMN2 (0.69) SMN1; SMN2GAALMNAGFERPOLB
SCHEMBL514571 0.77 SMN1; SMN2 (0.69) SMN1; SMN2POLBMAPTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140772-A1 COMPOSITION AND METHOD FOR INHIBITING RADICAL POLYMERISATION OF ETHYLENICALLY UNSATURATED ALIPHATIC MONOMERS RHODIA CHIMIE (FR) 2001-10-10 EP claimed
WO-2000037412-A1 COMPOSITION AND METHOD FOR INHIBITING RADICAL POLYMERISATION OF ETHYLENICALLY UNSATURATED ALIPHATIC MONOMERS RHODIA CHIMIE (FR) 2000-06-29 WO claimed
EP-1140772-A1 COMPOSITION AND METHOD FOR INHIBITING RADICAL POLYMERISATION OF ETHYLENICALLY UNSATURATED ALIPHATIC MONOMERS RHODIA CHIMIE (FR) 2001-10-10 EP disclosed
WO-2000037412-A1 COMPOSITION AND METHOD FOR INHIBITING RADICAL POLYMERISATION OF ETHYLENICALLY UNSATURATED ALIPHATIC MONOMERS RHODIA CHIMIE (FR) 2000-06-29 WO disclosed