SCHEMBL7935004

SCHEMBL7935004

CC(C)C[C@@H](C(=O)NN)[C@@H](C(=O)OC(C)(C)C)C(/C=C/c1ccccc1)(CC(C)C)S(C)(=O)=O

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 5/20 0.37
PSMB5 P28074 2/20 0.36
CYP2C19 P33261 1/20 0.35
POLB P06746 5/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 7/20 0.33
MAPK1 P28482 3/20 0.33
KMT2A Q03164 3/20 0.33
ATM Q13315 2/20 0.33
NPSR1 Q6W5P4 6/20 0.32
RECQL P46063 2/20 0.32
TDP1 Q9NUW8 2/20 0.32
MEN1 O00255 2/20 0.32
REN P00797 1/20 0.32
ALDH1A1 P00352 1/20 0.32
NPR3 P17342 1/20 0.32
XBP1 P17861 1/20 0.32
LARS1 Q9P2J5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4481740 0.88 ADAM17 (0.46) ADAM17CYP2C19LARS1
SCHEMBL6942610 0.88 ADAM17 (0.46) ADAM17CYP2C19LARS1
SCHEMBL6944661 0.83 ADAM17 (0.34) ADAM17PSMB5CYP2C19POLBMAPT
SCHEMBL6939550 0.81 MMP1 (0.38) ADAM17PSMB5POLBGAAMAPT
SCHEMBL6986272 0.81 MAPT (0.34) ADAM17PSMB5CYP2C19POLBGAA
SCHEMBL6945999 0.81 ADAM17 (0.43) ADAM17CYP2C19
SCHEMBL6945409 0.81 ADAM17 (0.43) ADAM17CYP2C19
SCHEMBL6940038 0.81
SCHEMBL6941767 0.80 ADAM17 (0.46) ADAM17CYP2C19LARS1
SCHEMBL6946650 0.80 ADAM17 (0.36) ADAM17PSMB5POLBGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed